SCHEMBL9947091

SCHEMBL9947091

CNc1cc(N(C)C2CCSC2)c(C(=O)NC2CCC(C(F)(F)F)CC2)cc1N

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGES O14684 13/20 0.37
DPP4 P27487 1/20 0.32
KCNH2 Q12809 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
S100A4 P26447 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.30
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9946650 1.00 PTGES (0.37) PTGESDPP4KCNH2DPP7S100A4
SCHEMBL9944944 0.89 NPC1 (0.40) S100A4
SCHEMBL9946636 0.89 PTGES (0.44) PTGESS100A4ALDH1A1POLBHPGD
SCHEMBL9946603 0.79 PTGES (0.48) PTGESS100A4ALDH1A1POLB
SCHEMBL9947009 0.79 PTGES (0.48) PTGESS100A4ALDH1A1POLB
SCHEMBL9899130 0.79 PTGES (0.48) PTGESS100A4
SCHEMBL9899126 0.79 PTGES (0.48) PTGESS100A4
SCHEMBL9946737 0.79 PTGES (0.48) PTGES
SCHEMBL9899024 0.78 PTGES (0.48) PTGESS100A4
SCHEMBL9946827 0.78 PTGES (0.48) PTGESS100A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076673-A1 6-AMINO-2-PHENYLAMINO-1H-BENZIMIDAZOLE-5-CARBOXAMIDE- DERIVATIVES AND THEIR USE AS MICROSOMAL PROSTAGLANDIN E2 SYNTHASE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 WO disclosed