SCHEMBL9952470

SCHEMBL9952470

COC(=O)c1ccc(-n2cc(-c3nn(C(=O)O)c4ccc(CBr)cc34)nn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.42
PSMD10 O75832 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK10 P53779 1/20 0.36
AURKA O14965 2/20 0.35
STIM1 Q13586 2/20 0.35
ORAI1 Q96D31 2/20 0.35
AURKB Q96GD4 1/20 0.35
S1PR1 P21453 1/20 0.35
RAB9A P51151 2/20 0.34
GAA P10253 1/20 0.34
SNCA P37840 1/20 0.34
NPC1 O15118 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ELANE P08246 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9951836 0.89 GRM1 (0.38) DHODHPSMD10AURKAAURKBS1PR1
SCHEMBL9952549 0.81 MEN1 (0.51) DHODHALDH1A1MAPK10POLB
SCHEMBL9952464 0.76 GRM1 (0.42) DHODHPSMD10AURKAAURKBPOLB
SCHEMBL10195459 0.72 MEN1 (0.46) DHODHS1PR1POLB
SCHEMBL19126510 0.67 PSMD10 (0.55) DHODHPSMD10AURKAAURKBNPC1
SCHEMBL9952570 0.66 GRM1 (0.40) ALDH1A1RAB9AGAANPC1SMN1; SMN2
SCHEMBL4050879 0.65 LOXL2 (0.63) ALDH1A1GAANPC1SMN1; SMN2
SCHEMBL31227601 0.64 PSMD10 (0.52) DHODHPSMD10ALDH1A1SMN1; SMN2POLB
SCHEMBL2671464 0.64 CA12 (0.45) ALDH1A1GAASMN1; SMN2POLBL3MBTL1
SCHEMBL33494 0.63 LOXL2 (0.66) ALDH1A1GAANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS Merck Serono S.A. (CH) 2013-10-30 EP disclosed
WO-2012084704-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO S.A. (CH) 2012-06-28 WO disclosed