SCHEMBL9953075

SCHEMBL9953075

COc1ncc(Br)cc1S(=O)(=O)NC1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 2/20 0.52
HTT P42858 4/20 0.51
TP53 P04637 1/20 0.50
CASP1 P29466 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.48
POLB P06746 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MAPK1 P28482 1/20 0.46
TSHR P16473 3/20 0.45
GAA P10253 3/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 2/20 0.45
ALDH1A1 P00352 4/20 0.45
MCOLN3 Q8TDD5 1/20 0.45
HPGD P15428 2/20 0.45
USP2 O75604 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PDE4A P27815 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954686 0.99 PIK3C3 (0.53) PIK3C3HTTTP53CASP1SMN1; SMN2
SCHEMBL14305926 0.96 PIK3C3 (0.55) PIK3C3HTTTP53CASP1SMN1; SMN2
SCHEMBL9954020 0.93 PIK3C3 (0.49) PIK3C3HTTTP53CASP1SMN1; SMN2
Pyridine SCHEMBL9955114 0.92 PIK3C3 (0.48) PIK3C3HTTTP53CASP1SMN1; SMN2
SCHEMBL21760960 0.88 PIK3C2G (0.48) PIK3C3HTTSMN1; SMN2POLBKDM4E
SCHEMBL19303684 0.88 PIK3C2G (0.48) PIK3C3HTTSMN1; SMN2POLBKDM4E
SCHEMBL9953196 0.88 PIK3CG (0.46) PIK3C3HTTTP53CASP1SMN1; SMN2
SCHEMBL9953667 0.81 PIK3C3 (0.42) PIK3C3POLBKDM4EHSD17B10MAPT
SCHEMBL14317987 0.80 PI4KB (0.42) PIK3C3SMN1; SMN2POLBALDH1A1MEN1
SCHEMBL23663187 0.79 PIK3C3 (0.47) PIK3C3HTTTP53CASP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed