SCHEMBL9954020

SCHEMBL9954020

COc1ncc(Br)cc1S(=O)(=O)NC1CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 2/20 0.49
KDM4E B2RXH2 1/20 0.49
HSD17B10 Q99714 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.42
HTT P42858 1/20 0.42
POLB P06746 2/20 0.41
TP53 P04637 1/20 0.41
CASP1 P29466 1/20 0.41
BRD4 O60885 2/20 0.41
BRD3 Q15059 2/20 0.41
PIK3C2G O75747 1/20 0.41
PIK3CG P48736 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
BRD2 P25440 1/20 0.41
SHMT2 P34897 1/20 0.40
OPRK1 P41145 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14305926 0.95 PIK3C3 (0.55) PIK3C3KDM4EHSD17B10L3MBTL1SMN1; SMN2
SCHEMBL9954686 0.95 PIK3C3 (0.53) PIK3C3KDM4EHSD17B10SMN1; SMN2HTT
SCHEMBL19303684 0.94 PIK3C2G (0.48) PIK3C3KDM4EHSD17B10L3MBTL1SMN1; SMN2
SCHEMBL21760960 0.94 PIK3C2G (0.48) PIK3C3KDM4EHSD17B10L3MBTL1SMN1; SMN2
SCHEMBL9953075 0.93 PIK3C3 (0.52) PIK3C3KDM4EHSD17B10SMN1; SMN2HTT
SCHEMBL9953196 0.91 PIK3CG (0.46) PIK3C3KDM4EHSD17B10L3MBTL1SMN1; SMN2
Pyridine SCHEMBL9955114 0.86 PIK3C3 (0.48) PIK3C3KDM4EHSD17B10SMN1; SMN2HTT
SCHEMBL9953667 0.85 PIK3C3 (0.42) PIK3C3KDM4EHSD17B10L3MBTL1POLB
SCHEMBL9953641 0.81 SHMT2 (0.44) L3MBTL1SMN1; SMN2POLBMEN1KMT2A
SCHEMBL23585301 0.80 L3MBTL1 (0.53) PIK3C3L3MBTL1SMN1; SMN2HTTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed