SCHEMBL9953472

SCHEMBL9953472

CNS(=O)(=O)c1cc(B2OC(C)(C)C(C)(C)O2)cnc1OC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.62
PIK3CD O00329 7/20 0.40
DGAT1 O75907 1/20 0.40
AAK1 Q2M2I8 1/20 0.39
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
CA12 O43570 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
CA14 Q9ULX7 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
PDGFRB P09619 1/20 0.34
KDR P35968 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL798817 0.88 ALPL (0.60) ALPLPIK3CDDGAT1AAK1CA1
SCHEMBL14317989 0.86 ALPL (0.59) ALPLPIK3CDDGAT1AAK1CA1
SCHEMBL9953660 0.86 ALPL (0.59) ALPLPIK3CDDGAT1AAK1CA1
SCHEMBL9954690 0.85 ALPL (0.57) ALPLPIK3CDDGAT1AAK1CA1
SCHEMBL9953730 0.84 ALPL (0.57) ALPLDGAT1AAK1L3MBTL1PIK3CG
SCHEMBL9953535 0.84 ALPL (0.57) ALPLPIK3CDDGAT1AAK1CA1
SCHEMBL14317975 0.84 ALPL (0.57) ALPLPIK3CDDGAT1AAK1CA1
SCHEMBL1502534 0.84 ALPL (0.56) ALPLDGAT1AAK1CA1CA2
SCHEMBL10288904 0.83 ALPL (0.56) ALPLPIK3CDDGAT1AAK1CA1
SCHEMBL9955177 0.83 ALPL (0.56) ALPLPIK3CDDGAT1AAK1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed