SCHEMBL9953566

SCHEMBL9953566

CC1OB(c2ccc3c(c2)CC(=O)N3)OC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.42
EPHX2 P34913 1/20 0.40
GRIA1 P42261 2/20 0.39
CACNG8 Q8WXS5 2/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37
PGR P06401 4/20 0.36
PDK2 Q15119 1/20 0.36
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
SMYD3 Q9H7B4 5/20 0.34
GAA P10253 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16230037 0.90 AHR (0.42) AHREPHX2GRIA1CACNG8PDE3B
SCHEMBL454535 0.81 AHR (0.49) AHREPHX2GRIA1CACNG8PDE3B
SCHEMBL31243804 0.81 AHR (0.49) AHREPHX2GRIA1CACNG8PDE3B
SCHEMBL16479504 0.78 MMP12 (0.50) PDE3BPDE3APGRGAAPKM
SCHEMBL12049915 0.74 AHR (0.42) AHREPHX2GRIA1CACNG8PDE3B
SCHEMBL392563 0.70 AHR (0.49) AHRPDK2
SCHEMBL30351303 0.70 AHR (0.49) AHRPDK2
SCHEMBL16812906 0.69 IDH1 (0.31)
SCHEMBL422134 0.69 PDE3B (0.44) PDE3BPDE3ACYP1A2CYP11B1CYP11B2
SCHEMBL17264079 0.68 LPL (0.48) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed