SCHEMBL9954787

SCHEMBL9954787

COc1ccc(CNc2nc3ccc(I)cc3c(=O)n2-c2cc(C)cc(C)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP3A4 P08684 2/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
GAA P10253 1/20 0.42
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953908 0.90 TP53 (0.47) MEN1KMT2ACYP3A4CA12CA1
SCHEMBL9954411 0.89 CA12 (0.44) MEN1KMT2ACYP3A4CA12CA1
SCHEMBL9954899 0.88 SMN1; SMN2 (0.47) MEN1KMT2ACYP3A4CA12CA1
SCHEMBL9953937 0.87 MEN1 (0.46) MEN1KMT2ACA12CA1CA2
SCHEMBL9955121 0.87 MAPT (0.46) MEN1KMT2ACYP3A4CYP1A2CYP2D6
SCHEMBL9953750 0.85 CYP3A4 (0.44) MEN1KMT2ACYP3A4CA12CA1
SCHEMBL9953016 0.85 CYP3A4 (0.44) MEN1KMT2ACYP3A4CA12CA1
SCHEMBL9953858 0.85 MEN1 (0.41) MEN1KMT2ACYP3A4CA12CA1
SCHEMBL9954815 0.85 ACP1 (0.47) CA12CA1CA2CA9
SCHEMBL9953860 0.85 CYP1A2 (0.42) MEN1KMT2ACYP3A4CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed