SCHEMBL9953908

SCHEMBL9953908

COc1ccc(CNc2nc3ccc(I)cc3c(=O)n2-c2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.47
LMNA P02545 1/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
HPGD P15428 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPT P10636 2/20 0.46
THRB P10828 1/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
GAA P10253 1/20 0.45
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954899 0.94 SMN1; SMN2 (0.47) TP53LMNAALDH1A1KDM4EMAPT
SCHEMBL9953937 0.91 MEN1 (0.46) TP53LMNAALDH1A1L3MBTL1MAPT
SCHEMBL9953858 0.91 MEN1 (0.41) TP53LMNAALDH1A1KDM4EHPGD
SCHEMBL9953860 0.91 CYP1A2 (0.42) TP53LMNAALDH1A1KDM4EHPGD
SCHEMBL9954787 0.90 MEN1 (0.44) TP53LMNACYP1A2CYP3A4CYP2D6
SCHEMBL9954411 0.89 CA12 (0.44) TP53LMNAALDH1A1MAPTTHRB
SCHEMBL9953429 0.89 TP53 (0.45) TP53LMNAMAPTTHRBCYP1A2
SCHEMBL9954480 0.89 L3MBTL1 (0.46) TP53LMNAALDH1A1KDM4EHPGD
SCHEMBL9954815 0.89 ACP1 (0.47) CA12CA1CA2CA9ACP1
SCHEMBL9955556 0.89 CA12 (0.47) ALDH1A1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed