SCHEMBL9954967

SCHEMBL9954967

CC(C)(C)C(=O)N1CCc2nc(S(C)(=O)=O)ncc2C1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.46
RIPK1 Q13546 2/20 0.42
HDAC6 Q9UBN7 3/20 0.40
HDAC8 Q9BY41 1/20 0.40
HSP90AA1 P07900 5/20 0.39
HSP90AB1 P08238 4/20 0.39
ENPP2 Q13822 1/20 0.39
HSP90B1 P14625 1/20 0.38
PDK2 Q15119 1/20 0.38
PDGFRB P09619 1/20 0.38
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL785054 0.86 MAPT (0.43) MAPTHSP90AA1HSP90AB1ENPP2HSP90B1
SCHEMBL786189 0.84 MAPT (0.65) MAPTENPP2PDGFRB
SCHEMBL14496905 0.77 CYP2C19 (0.40) MAPT
SCHEMBL2246755 0.76 ESR1 (0.41) MAPT
SCHEMBL1503713 0.76 HSP90AA1 (0.38) MAPTHSP90AA1HSP90B1
SCHEMBL741206 0.75 MAPT (0.51) MAPT
SCHEMBL16870041 0.70 MAPT (0.33) MAPT
SCHEMBL15309369 0.70 ABHD6 (0.48) RIPK1HDAC6HDAC8HSP90AA1PDK2
SCHEMBL18818957 0.69 TP53 (0.33) MAPT
SCHEMBL24921008 0.69 HTR6 (0.36) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085167-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO disclosed