SCHEMBL9956286

SCHEMBL9956286

Cc1cccc(-c2co[c]n2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP3 O14638 2/20 0.45
IDO1 P14902 1/20 0.45
METAP2 P50579 1/20 0.45
RAB9A P51151 6/20 0.42
NPC1 O15118 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
HPGD P15428 2/20 0.42
TSHR P16473 1/20 0.42
KMO O15229 2/20 0.40
KDM4E B2RXH2 1/20 0.40
XDH P47989 1/20 0.40
ALDH1A1 P00352 3/20 0.39
NFKB1 P19838 2/20 0.39
NFKB2 Q00653 2/20 0.39
RELA Q04206 2/20 0.39
ACHE P22303 2/20 0.39
BCHE P06276 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 1/20 0.39
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9955620 0.79 IDO1 (0.45) IDO1RAB9ANPC1SMN1; SMN2KMO
SCHEMBL9956598 0.79 IDO1 (0.45) IDO1RAB9ANPC1SMN1; SMN2TSHR
SCHEMBL2092720 0.77 ENPP3 (0.46) ENPP3METAP2RAB9ANPC1SMN1; SMN2
SCHEMBL102449 0.77 RAB9A (0.41) IDO1METAP2RAB9ANPC1SMN1; SMN2
SCHEMBL9488955 0.76 NPC1 (0.40) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL8123490 0.76 IDO1 (0.35) IDO1RAB9ANPC1SMN1; SMN2KDM4E
SCHEMBL17028965 0.75 IDO1 (0.49) IDO1RAB9AHPGDKMOKDM4E
SCHEMBL1894497 0.71 MAOB (0.37) KDM4EALDH1A1MAPT
SCHEMBL3629467 0.70 IDO1 (0.55) ENPP3IDO1METAP2RAB9ANPC1
SCHEMBL11674446 0.69 RAB9A (0.47) ENPP3IDO1METAP2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed