SCHEMBL9957714

SCHEMBL9957714

Cc1c(O)cccc1C(=N)Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.48
ATM Q13315 1/20 0.48
HSD17B1 P14061 3/20 0.39
HSD17B2 P37059 3/20 0.39
LMNA P02545 4/20 0.35
HSD17B10 Q99714 4/20 0.35
ALDH1A1 P00352 4/20 0.35
HPGD P15428 4/20 0.35
TP53 P04637 3/20 0.35
KDM4E B2RXH2 3/20 0.35
ALOX15 P16050 2/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
ALOX12 P18054 1/20 0.35
MAPK1 P28482 1/20 0.35
TSHR P16473 4/20 0.35
NPC1 O15118 2/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
CA1 P00915 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23550094 0.80 TRPA1 (0.50) TRPA1ATMHSD17B1HSD17B2LMNA
SCHEMBL4976492 0.78 TRPA1 (0.48) TRPA1ATMHSD17B1HSD17B2LMNA
SCHEMBL28171956 0.78 TRPA1 (0.48) TRPA1ATMHSD17B1HSD17B2LMNA
SCHEMBL27303906 0.78 TRPA1 (0.54) TRPA1ATMHSD17B1HSD17B2LMNA
SCHEMBL2134038 0.77 TRPA1 (0.46) TRPA1ATMHSD17B1HSD17B2LMNA
SCHEMBL4711338 0.77 HPGD (0.48) LMNAHSD17B10ALDH1A1HPGDTP53
SCHEMBL30525835 0.77 HPGD (0.48) LMNAHSD17B10ALDH1A1HPGDTP53
SCHEMBL16951421 0.75 TRPA1 (0.54) TRPA1ATMHSD17B1HSD17B2LMNA
SCHEMBL2928032 0.74 HSD17B14 (0.38) HSD17B1HSD17B2LMNAHSD17B10ALDH1A1
SCHEMBL20168228 0.74 CA1 (0.46) LMNAHSD17B10ALDH1A1HPGDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105061313-B Androgen receptor modulating compounds 奥赖恩公司 2017-07-18 CN disclosed
EP-2655370-A1 COMPOSITIONS AND METHODS FOR MODULATING FXR IRM LLC (BM) 2013-10-30 EP disclosed
WO-2012087519-A1 COMPOSITIONS AND METHODS FOR MODULATING FXR IRM LLC (BM) 2012-06-28 WO disclosed