SCHEMBL995788

SCHEMBL995788

COc1cc(OC)c(C(=O)/C=C/c2cccc(Cl)c2)cc1SC

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.51
AR P10275 2/20 0.50
MAOB P27338 2/20 0.50
MAOA P21397 1/20 0.50
CXCL12 P48061 5/20 0.48
ABCG2 Q9UNQ0 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
MAPT P10636 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
CYP1A1 P04798 1/20 0.46
CYP1B1 Q16678 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL995789 1.00 ABCB1 (0.51) ABCB1ARMAOBMAOACXCL12
SCHEMBL996603 0.95 AR (0.50) ABCB1ARMAOBMAOACXCL12
SCHEMBL996606 0.95 AR (0.50) ABCB1ARMAOBMAOACXCL12
SCHEMBL996233 0.90 ABCB1 (0.47) ABCB1ARMAOBMAOACXCL12
SCHEMBL996235 0.90 ABCB1 (0.47) ABCB1ARMAOBMAOACXCL12
SCHEMBL996825 0.87 ABCG2 (0.64) ARMAOBMAOACXCL12ABCG2
SCHEMBL996824 0.87 ABCG2 (0.64) ARMAOBMAOACXCL12ABCG2
SCHEMBL997192 0.87 MAPT (0.62) MAOBMAOAABCG2CYP1A2CYP3A4
SCHEMBL997194 0.87 MAPT (0.62) MAOBMAOAABCG2CYP1A2CYP3A4
SCHEMBL997861 0.83 PDE4A (0.64) ARMAOBABCG2CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO claimed
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO disclosed