SCHEMBL996235

SCHEMBL996235

COc1cc(OCC(=O)O)c(C(=O)C=Cc2cccc(Cl)c2)cc1SC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.47
MAOB P27338 2/20 0.46
MAOA P21397 1/20 0.46
CYSLTR2 Q9NS75 2/20 0.46
CYSLTR1 Q9Y271 2/20 0.46
AR P10275 2/20 0.43
MEN1 O00255 2/20 0.43
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
NR1I2 O75469 1/20 0.42
LMNA P02545 1/20 0.42
PGR P06401 1/20 0.42
ADRB2 P07550 1/20 0.42
ADRB1 P08588 1/20 0.42
ADORA3 P0DMS8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL996233 1.00 ABCB1 (0.47) ABCB1MAOBMAOACYSLTR2CYSLTR1
SCHEMBL997652 0.90 MAPT (0.54) CYSLTR1MEN1MAPTKMT2ANPC1
SCHEMBL997653 0.90 MAPT (0.54) CYSLTR1MEN1MAPTKMT2ANPC1
SCHEMBL995788 0.90 ABCB1 (0.51) ABCB1MAOBMAOAARMEN1
SCHEMBL995789 0.90 ABCB1 (0.51) ABCB1MAOBMAOAARMEN1
SCHEMBL996606 0.85 AR (0.50) ABCB1MAOBMAOAARMEN1
SCHEMBL996603 0.85 AR (0.50) ABCB1MAOBMAOAARMEN1
SCHEMBL996875 0.85 ABCG2 (0.56) CYSLTR2CYSLTR1MEN1MAPTKMT2A
SCHEMBL996877 0.85 ABCG2 (0.56) CYSLTR2CYSLTR1MEN1MAPTKMT2A
SCHEMBL996701 0.83 ABCG2 (0.56) ABCB1MAOBCYSLTR1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO disclosed