SCHEMBL997192

SCHEMBL997192

COc1cc(OC)c(C(=O)/C=C/c2ccccc2)cc1SC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.62
KMT2A Q03164 3/20 0.62
NPC1 O15118 2/20 0.62
RAB9A P51151 2/20 0.62
MEN1 O00255 2/20 0.62
ABCG2 Q9UNQ0 5/20 0.56
NPSR1 Q6W5P4 2/20 0.55
CYP1A1 P04798 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP1B1 Q16678 1/20 0.55
TNFRSF1A P19438 3/20 0.54
ATM Q13315 2/20 0.52
LMNA P02545 1/20 0.52
RECQL P46063 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
CAPN1 P07384 1/20 0.51
PARP1 P09874 1/20 0.51
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
KCNA3 P22001 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL997194 1.00 MAPT (0.62) MAPTKMT2ANPC1RAB9AMEN1
SCHEMBL997735 0.95 MAPT (0.62) MAPTKMT2ANPC1RAB9AMEN1
SCHEMBL997734 0.95 MAPT (0.62) MAPTKMT2ANPC1RAB9AMEN1
SCHEMBL997653 0.90 MAPT (0.54) MAPTKMT2ANPC1RAB9AMEN1
SCHEMBL997652 0.90 MAPT (0.54) MAPTKMT2ANPC1RAB9AMEN1
SCHEMBL997364 0.88 ABCG2 (0.67) MAPTKMT2ANPC1RAB9AMEN1
SCHEMBL997363 0.88 ABCG2 (0.67) MAPTKMT2ANPC1RAB9AMEN1
SCHEMBL996824 0.87 ABCG2 (0.64) MAPTABCG2TNFRSF1ACAPN1PARP1
SCHEMBL996825 0.87 ABCG2 (0.64) MAPTABCG2TNFRSF1ACAPN1PARP1
SCHEMBL995788 0.87 ABCB1 (0.51) MAPTKMT2ANPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO claimed
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO disclosed