SCHEMBL995823

SCHEMBL995823

NC(=O)c1ccccc1-c1cccc2ncccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.52
NSD2 O96028 1/20 0.49
PARP1 P09874 1/20 0.49
PDE4B Q07343 1/20 0.48
CSNK1A1 P48729 1/20 0.48
TYRO3 Q06418 1/20 0.48
DYRK1B Q9Y463 1/20 0.48
PABPC1 P11940 2/20 0.47
EIF4H Q15056 2/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
BCAT2 O15382 1/20 0.46
KDM4E B2RXH2 2/20 0.45
SLC22A12 Q96S37 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30863578 1.00 NUDT1 (0.52) NUDT1NSD2PARP1PDE4BCSNK1A1
SCHEMBL27991327 0.92 NUDT1 (0.61) NUDT1CSNK1A1TYRO3DYRK1BBCAT2
SCHEMBL31032078 0.86 PARP1 (0.47) NSD2PARP1PDE4BPABPC1EIF4H
SCHEMBL17559805 0.86 NSD2 (0.54) NSD2PABPC1EIF4HKDM4ESLC22A12
SCHEMBL1804352 0.85 PARP1 (0.56) NSD2PARP1PDE4BPABPC1EIF4H
SCHEMBL8221166 0.85 PARP1 (0.56) NSD2PARP1PDE4BPABPC1EIF4H
SCHEMBL30646218 0.83 BCAT2 (0.63) NUDT1PARP1CSNK1A1TYRO3DYRK1B
SCHEMBL27872261 0.81 NUDT1 (0.59) NUDT1PARP1CSNK1A1TYRO3DYRK1B
Quinoline SCHEMBL28140561 0.81 PARP1 (0.57) NSD2PARP1PDE4BPABPC1EIF4H
SCHEMBL7502767 0.79 NUDT1 (0.48) NUDT1PARP1PDE4BKDM4ESLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011011514-A1 HETEROARYL BENZAMIDES, COMPOSITIONS AND METHODS OF USE THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2011-01-27 WO claimed
CN-100393720-C Cyclic benzimidazoles. ALTANA PHARMA AG (DE) 2008-06-11 CN claimed
WO-2011011514-A1 HETEROARYL BENZAMIDES, COMPOSITIONS AND METHODS OF USE THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2011-01-27 WO disclosed
CN-100393720-C Cyclic benzimidazoles. ALTANA PHARMA AG (DE) 2008-06-11 CN disclosed
CN-1764662-A Cyclic benzimidazoles. ALTANA PHARMA AG (DE) 2006-04-26 CN disclosed