SCHEMBL9958370

SCHEMBL9958370

CC(C)(C)c1ccc(CNCCc2cc(C(F)(F)F)ccn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.47
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
SCN8A Q9UQD0 2/20 0.43
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
PHGDH O43175 1/20 0.37
ADRB2 P07550 1/20 0.37
MITF O75030 1/20 0.37
GAA P10253 1/20 0.37
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576790 0.82 CA1 (0.47) CA1CA2SCN8AKMT2AKDM4E
SCHEMBL5176818 0.79 CA1 (0.62) CA1CA2SCN8AKMT2AGAA
SCHEMBL13778175 0.79 ALDH1A1 (0.56) CA1CA2KMT2AKDM4EMITF
SCHEMBL3235999 0.77 KDM4E (0.58) ROCK1CA1CA2SCN8AKMT2A
SCHEMBL5175994 0.76 CA1 (0.47) CA1CA2SCN8AKMT2A
SCHEMBL3580858 0.74 CA1 (0.48) ROCK1CA1CA2SCN8AKMT2A
SCHEMBL3244176 0.74 CA1 (0.50) ROCK1CA1CA2KMT2AKDM4E
SCHEMBL47299 0.74 CA1 (0.50) ROCK1CA1CA2SCN8AKMT2A
SCHEMBL20902780 0.74 CA1 (0.71) CA1CA2KMT2AGAA
SCHEMBL24258324 0.74 SIRT2 (0.43) SCN8AADRB2GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed