SCHEMBL9958985

SCHEMBL9958985

CCCCN(C)C(=O)C1C(=O)N(O)C(=O)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
TSHR P16473 3/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 2/20 0.37
CYP1A2 P05177 1/20 0.37
HPGD P15428 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9959015 0.82 MEN1 (0.49) KDM4ETSHRKMT2AALDH1A1MEN1
SCHEMBL9959279 0.80 KDM4E (0.44) KDM4ETSHRKMT2AALDH1A1MEN1
SCHEMBL10154016 0.77 MEN1 (0.38) KDM4EKMT2AALDH1A1MEN1L3MBTL1
SCHEMBL10153314 0.77 KMT2A (0.54) KDM4ETSHRKMT2AALDH1A1MEN1
SCHEMBL10153707 0.76 KMT2A (0.55) KDM4EKMT2AALDH1A1MEN1GAA
SCHEMBL19380275 0.75 ALDH1A1 (0.42) KMT2AALDH1A1MEN1CYP1A2HPGD
SCHEMBL31653849 0.75 ALDH1A1 (0.42) KMT2AALDH1A1MEN1CYP1A2HPGD
SCHEMBL9952553 0.75 KMT2A (0.54) KDM4EKMT2AALDH1A1MEN1GAA
SCHEMBL9952669 0.75 KMT2A (0.54) KDM4EKMT2AALDH1A1MEN1GAA
SCHEMBL9959705 0.75 KMT2A (0.54) KDM4EKMT2AALDH1A1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed