Histidine

Histidine

SCHEMBL995910

NC(Cc1c[nH]cn1)C(=O)O.N[C@@H](Cc1c[nH]cn1)C(=O)O

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP1A2 P05177 1/20 0.46
PKM P14618 2/20 0.43
ALPI P09923 1/20 0.43
PTGS1 P23219 1/20 0.43
XIAP P98170 1/20 0.43
GRIA2 P42262 5/20 0.41
GRIA1 P42261 4/20 0.41
GRIA3 P42263 4/20 0.41
GRIA4 P48058 4/20 0.41
HSD17B10 Q99714 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
BLM P54132 2/20 0.40
PMP22 Q01453 2/20 0.40
KMT2A Q03164 2/20 0.40
HIF1A Q16665 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Histidine SCHEMBL8316642 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL8080341 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL388561 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL18824897 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL388563 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL3258 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL163443 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL3259 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL163442 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI
Histidine SCHEMBL29500208 1.00 SLC7A5 (0.47) SLC7A5CYP3A4CYP1A2PKMALPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465973-B1 PLATING CATALYST AND METHOD ROHM & HAAS ELECT MAT (US) 2018-11-28 EP disclosed
EP-3233136-A1 TARGETED GAS-FILLED MICROVESICLES FORMULATION Bracco Suisse SA (CH) 2017-10-25 EP disclosed
WO-2016097130-A1 TARGETED GAS-FILLED MICROVESICLES FORMULATION BRACCO SUISSE SA (CH) 2016-06-23 WO disclosed
US-9234282-B2 Plating catalyst and method ROHM AND HAAS ELECTRONIC MATERIALS LLC (US) 2016-01-12 US disclosed
US-20140083860-A1 PLATING CATALYST AND METHOD ROHM AND HAAS ELECTRONIC MATERIALS LLC 2014-03-27 US disclosed
US-8591637-B2 Plating catalyst and method ROHM AND HAAS ELECTRONIC MATERIALS LLC (US) 2013-11-26 US disclosed
EP-2566501-A2 METHOD AND DEVICE FOR TRANSDERMAL DELIVERY OF PARATHYROID HORMONE USING A MICROPROJECTION ARRAY Corium International, Inc. (US) 2013-03-13 EP disclosed
EP-2465973-A2 Plating catalyst and method Rohm and Haas Electronic Materials LLC (US) 2012-06-20 EP disclosed
US-20120145555-A1 PLATING CATALYST AND METHOD ROHM AND HAAS ELECTRONIC MATERIALS LLC (US) 2012-06-14 US disclosed
EP-2449488-A1 METHOD FOR NORMALIZATION IN METABOLOMICS ANALYSIS METHODS WITH ENDOGENOUS REFERENCE METABOLITES BIOCRATES Life Sciences AG (AT) 2012-05-09 EP disclosed
WO-2011140274-A2 METHOD AND DEVICE FOR TRANSDERMAL DELIVERY OF PARATHYROID HORMONE USING A MICROPROJECTION ARRAY CORIUM INTERNATIONAL, INC. (US) 2011-11-10 WO disclosed
WO-2011000753-A1 METHOD FOR NORMALIZATION IN METABOLOMICS ANALYSIS METHODS WITH ENDOGENOUS REFERENCE METABOLITES BIOCRATES LIFE SCIENCES AG (AT) 2011-01-06 WO disclosed
EP-0806947-A4 FORMULATIONS AND METHODS FOR REDUCING SKIN IRRITATION COSMEDERM TECHNOLOGIES (US) 1998-10-14 EP disclosed
EP-0806947-A1 FORMULATIONS AND METHODS FOR REDUCING SKIN IRRITATION COSMEDERM TECHNOLOGIES (US) 1997-11-19 EP disclosed
WO-1996023490-A9 FORMULATIONS AND METHODS FOR REDUCING SKIN IRRITATION 1996-12-27 WO disclosed
WO-1996023490-A1 FORMULATIONS AND METHODS FOR REDUCING SKIN IRRITATION COSMEDERM TECHNOLOGIES (US) 1996-08-08 WO disclosed