SCHEMBL9959585

SCHEMBL9959585

O=C(O)NC1CCCC(Cn2ncc3ccccc32)C1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
TSHR P16473 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CRHR1 P34998 1/20 0.48
KMO O15229 1/20 0.46
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
RECQL P46063 1/20 0.41
CFD P00746 1/20 0.41
POLB P06746 2/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10237675 0.84 L3MBTL1 (0.48) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL31429406 0.81 RECQL (0.51) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL25741023 0.80 CHRM2 (0.49) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL3904701 0.77 DRD2 (0.52) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL25740903 0.76 CHRM2 (0.48) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL25740899 0.76 CHRM2 (0.48) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL9960182 0.76 CHRM2 (0.46) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL15284866 0.76 NPC1 (0.47) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL15284867 0.76 NPC1 (0.47) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1
SCHEMBL5946285 0.75 RECQL (0.54) NPC1RAB9ASMN1; SMN2TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2654748-A1 INDAZOLE DERIVATIVES USEFUL AS ERK INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-10-30 EP disclosed
WO-2012087772-A1 INDAZOLE DERIVATIVES USEFUL AS ERK INHIBITORS SCHERING CORPORATION (US) 2012-06-28 WO disclosed