SCHEMBL9959773

SCHEMBL9959773

O=C(NCc1ccc(F)cc1)C1C(=O)N(O)C(=O)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
L3MBTL1 Q9Y468 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
ALDH1A1 P00352 4/20 0.41
MAPT P10636 3/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PRMT5 O14744 3/20 0.39
WDR77 Q9BQA1 3/20 0.39
CASP6 P55212 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29418268 1.00 GAA (0.47) GAAL3MBTL1MEN1KMT2AMAOA
SCHEMBL19380302 0.87 ALDH1A1 (0.48) GAAMEN1KMT2AALDH1A1MAPT
SCHEMBL30675135 0.87 PRMT5 (0.47) L3MBTL1MEN1KMT2AALDH1A1LMNA
SCHEMBL29411937 0.83 CNR1 (0.45) ALDH1A1RAB9APRMT5WDR77
SCHEMBL30499662 0.83 ALDH1A1 (0.41) L3MBTL1MEN1KMT2AALDH1A1LMNA
SCHEMBL9958767 0.83 CNR1 (0.45) ALDH1A1RAB9APRMT5WDR77
SCHEMBL9959490 0.83 PRMT5 (0.42) L3MBTL1MEN1KMT2AALDH1A1LMNA
SCHEMBL9959238 0.83 ALDH1A1 (0.41) L3MBTL1MEN1KMT2AALDH1A1LMNA
SCHEMBL29696849 0.82 NPC1 (0.47) L3MBTL1MEN1KMT2AALDH1A1MAPT
SCHEMBL9953409 0.81 POLB (0.50) ALDH1A1RAB9ASMN1; SMN2PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed