SCHEMBL997653

SCHEMBL997653

COc1cc(OCC(=O)O)c(C(=O)C=Cc2ccccc2)cc1SC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
LMNA P02545 2/20 0.49
NR1I2 O75469 1/20 0.49
PGR P06401 1/20 0.49
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
HPGD P15428 1/20 0.49
CNR1 P21554 1/20 0.49
TBXA2R P21731 1/20 0.49
SLC6A2 P23975 1/20 0.49
AGTR1 P30556 1/20 0.49
ADRA1A P35348 1/20 0.49
OPRD1 P41143 1/20 0.49
OPRK1 P41145 1/20 0.49
BLM P54132 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL997652 1.00 MAPT (0.54) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL996875 0.92 ABCG2 (0.56) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL996877 0.92 ABCG2 (0.56) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL999702 0.90 MAPT (0.49) MAPTMEN1KMT2ALMNANR1I2
SCHEMBL999701 0.90 MAPT (0.49) MAPTMEN1KMT2ALMNANR1I2
SCHEMBL996233 0.90 ABCB1 (0.47) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL996235 0.90 ABCB1 (0.47) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL997194 0.90 MAPT (0.62) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL997192 0.90 MAPT (0.62) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL996701 0.86 ABCG2 (0.56) MAPTMEN1KMT2ALMNAABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO disclosed