SCHEMBL9963570

SCHEMBL9963570

Cc1c2nc(NCC(=O)N3CCCC3)sc2cc2sc(NC(=O)CN(C)C)nc12

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.41
ACHE P22303 3/20 0.39
P2RX7 Q99572 2/20 0.39
GRIN2B Q13224 1/20 0.38
ITK Q08881 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
ACP1 P24666 1/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 3/20 0.36
PRMT3 O60678 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9963559 0.86 PTGS2 (0.40) PTGS2ITKALDH1A1HPGDPRMT3
SCHEMBL9963539 0.85 PTGS2 (0.43) PTGS2ALDH1A1HPGDPRMT3LMNA
SCHEMBL9963695 0.84 PTGS2 (0.49) PTGS2ALDH1A1HPGDMAPTPRMT3
SCHEMBL9963577 0.84 PTGS2 (0.44) PTGS2ALDH1A1HPGDNPC1MAPT
SCHEMBL9963632 0.83 PTGS2 (0.40) PTGS2ACHEP2RX7GRIN2BALDH1A1
SCHEMBL9963581 0.83 PTGS2 (0.42) PTGS2ACHEP2RX7GRIN2BALDH1A1
SCHEMBL9963593 0.83 PTGS2 (0.46) PTGS2ALDH1A1HPGDMAPTPRMT3
SCHEMBL9963545 0.83 PTGS2 (0.51) PTGS2ALDH1A1HPGDMAPTPRMT3
SCHEMBL9963588 0.82 ACHE (0.46) PTGS2ACHEP2RX7GRIN2BALDH1A1
SCHEMBL9963484 0.82 PTGS2 (0.45) PTGS2ALDH1A1HPGDPRMT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2032583-B1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2014-11-19 EP disclosed
US-8203001-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-19 US disclosed
US-8203001-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-19 US disclosed
US-20090258857-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-15 US disclosed
US-20090258857-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-15 US disclosed
WO-2007144370-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-12-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090258857-A1 CHEMICAL COMPOUNDS CCNA1, CCNT1, MKI67 PTGS2 2872/4885ACHE 1479/4885P2RX7 1644/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.