SCHEMBL9965164

SCHEMBL9965164

C=N/C=C\N(N)c1ccc(C(F)(F)F)cc1NC(=O)Nc1ccc(-n2c[n+]([O-])c(C(N)=O)c2N)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 0.37
CA12 O43570 3/20 0.37
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA9 Q16790 3/20 0.37
PDGFRB P09619 2/20 0.34
EPHA3 P29320 1/20 0.34
EPHB4 P54760 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KIT P10721 1/20 0.33
FLT3 P36888 1/20 0.33
EPHX2 P34913 1/20 0.32
IDO1 P14902 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4264162 0.75 ALDH1A1 (0.49) KDRCA12CA1CA2CA9
SCHEMBL4260344 0.74 KDR (0.56) KDRCA12CA1CA2CA9
SCHEMBL4259334 0.74 IDH2 (0.50) KDRCA12CA1CA2CA9
SCHEMBL5444130 0.62 KDR (0.57) KDRCA12CA1CA2CA9
SCHEMBL5445047 0.59 RAF1 (0.51) KDRPDGFRBMAPT
SCHEMBL2335664 0.59 ALDH1A1 (0.52) KDRMEN1KMT2AMAPT
SCHEMBL5440844 0.58 CA12 (0.53) KDRCA12CA1CA2CA9
SCHEMBL5439135 0.58 KDR (0.52) KDRCA12CA1CA2CA9
SCHEMBL5441043 0.57 CA12 (0.53) KDRCA12CA1CA2CA9
SCHEMBL5436578 0.56 KDR (0.64) KDRPDGFRBEPHA3EPHB4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082746-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-06-21 WO disclosed