SCHEMBL9965286

SCHEMBL9965286

Cc1cc2c(N)ccc(C)c2nc1Nc1cc(C(F)(F)F)ccn1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SYK P43405 6/20 0.42
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TEAD1 P28347 1/20 0.39
MAP3K12 Q12852 3/20 0.38
IDH2 P48735 1/20 0.38
BRAF P15056 1/20 0.37
AURKA O14965 2/20 0.35
RPS6KB1 P23443 1/20 0.35
RIPK2 O43353 1/20 0.35
KDR P35968 1/20 0.35
MAPK14 Q16539 1/20 0.35
MAPK1 P28482 1/20 0.35
TAS2R14 Q9NYV8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9938726 0.90 SYK (0.40) SYKNOS3NOS2ALDH1A1GAA
SCHEMBL9972399 0.83 IDH2 (0.41) SYKNOS3NOS2ALDH1A1GAA
SCHEMBL25894573 0.74 SYK (0.38) SYKALDH1A1GAAL3MBTL1TEAD1
SCHEMBL17443159 0.73 IDH2 (0.45) SYKNOS3NOS2ALDH1A1GAA
SCHEMBL20124507 0.73 SYK (0.37) SYKALDH1A1GAAL3MBTL1TEAD1
SCHEMBL9965317 0.71 NOS3 (0.42) SYKNOS3NOS2ALDH1A1L3MBTL1
SCHEMBL9943626 0.71 ALDH1A1 (0.42) SYKALDH1A1GAAL3MBTL1TEAD1
SCHEMBL22135110 0.69 IDH2 (0.38) SYKALDH1A1GAAL3MBTL1TEAD1
SCHEMBL9939354 0.69 MAPK10 (0.44) SYKALDH1A1GAAL3MBTL1MAP3K12
SCHEMBL9943489 0.67 CLK1 (0.40) SYKALDH1A1GAAL3MBTL1IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012080953-A1 COMPOUNDS USEFUL FOR TREATING AIDS SPLICOS (FR) 2012-06-21 WO disclosed