SCHEMBL9965448

SCHEMBL9965448

Cc1ccc(-c2ccccc2NC2CCN(C=O)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.42
DRD2 P14416 1/20 0.39
LMNA P02545 2/20 0.39
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
IDO1 P14902 1/20 0.38
MCHR1 Q99705 1/20 0.37
TSHR P16473 2/20 0.36
CHRM3 P20309 1/20 0.36
ACHE P22303 2/20 0.35
BCHE P06276 1/20 0.35
MAPK3 P27361 1/20 0.35
NPC1 O15118 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14639693 0.86 CHRM3 (0.42) BRD4DRD2KMT2ACHRM3ACHE
SCHEMBL9965478 0.82 TSHR (0.46) BRD4LMNAALDH1A1MEN1KMT2A
SCHEMBL14141237 0.72 MAPK3 (0.44) BRD4ALDH1A1KMT2ATSHRMAPK3
SCHEMBL13801296 0.71 MAPK3 (0.46) BRD4MEN1KMT2ATSHRMAPK3
SCHEMBL9965473 0.71 TSHR (0.54) BRD4ALDH1A1MEN1KMT2AATM
SCHEMBL29127243 0.70 ALDH1A1 (0.49) LMNAALDH1A1MEN1KMT2AATM
SCHEMBL10224761 0.70 TSHR (0.45) BRD4ALDH1A1MEN1KMT2AATM
SCHEMBL9965412 0.70 MLNR (0.47) LMNAALDH1A1KMT2ATSHRCHRM3
SCHEMBL9965418 0.70 HDAC3 (0.48) ALDH1A1TSHRCHRM3CYP3A4MAPT
SCHEMBL27927468 0.70 CARM1 (0.51) BRD4CA12CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-B1 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS STERIX LTD (GB) 2012-06-20 EP disclosed