SCHEMBL14141237

SCHEMBL14141237

CC(=O)Nc1ccccc1NC1CCN(C=O)CC1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK3 P27361 2/20 0.44
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
BRD4 O60885 1/20 0.41
MAPK1 P28482 1/20 0.41
MAPT P10636 1/20 0.40
TSHR P16473 2/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SLC18A3 Q16572 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13801296 0.88 MAPK3 (0.46) MAPK3BRD4MAPK1MAPTTSHR
SCHEMBL22605778 0.85 ALDH1A1 (0.45) ALDH1A1HPGDMAPK1MAPTTSHR
SCHEMBL5365015 0.75 SLC18A3 (0.49) ALDH1A1TSHRSMN1; SMN2CYP1A2CYP2D6
SCHEMBL6152397 0.75 SLC18A3 (0.49) ALDH1A1TSHRSMN1; SMN2CYP1A2CYP2D6
SCHEMBL13801304 0.73 BRD4 (0.39) MAPK3ALDH1A1BRD4MAPK1KMT2A
SCHEMBL5857181 0.73 KDM4E (0.47) ALDH1A1
SCHEMBL28537777 0.73 FNTA (0.46) ALDH1A1POLBCYP1A2CYP3A4CYP2D6
SCHEMBL9965448 0.72 BRD4 (0.42) MAPK3ALDH1A1BRD4MAPTTSHR
SCHEMBL27766517 0.72 SMN1; SMN2 (0.44) MAPK3ALDH1A1MAPK1MAPTHTT
SCHEMBL6689158 0.72 ALDH1A1 (0.74) ALDH1A1HPGDMAPK1TSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440976-B1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production BOEHRINGER INGELHEIM PHARMA (DE) 2008-07-23 EP disclosed