SCHEMBL9965449

SCHEMBL9965449

CC(=O)N1CCC(Nc2ccccc2Cc2ccc(Cl)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
NSD2 O96028 1/20 0.47
ALDH1A1 P00352 2/20 0.46
LMNA P02545 2/20 0.46
HRH1 P35367 1/20 0.45
KMT2A Q03164 1/20 0.45
CCR3 P51677 1/20 0.44
BRD4 O60885 1/20 0.43
MAPT P10636 1/20 0.43
EPHX2 P34913 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
MAPK3 P27361 1/20 0.42
HPGD P15428 1/20 0.42
UBE2M P61081 1/20 0.42
DCUN1D1 Q96GG9 1/20 0.42
GLA P06280 1/20 0.41
TSHR P16473 1/20 0.41
RORC P51449 1/20 0.41
ALOX12 P18054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965476 0.81 HRH1 (0.42) KDM4ESMN1; SMN2ALDH1A1LMNAHRH1
SCHEMBL9965421 0.80 NSD2 (0.54) KDM4ENSD2ALDH1A1KMT2ABRD4
SCHEMBL10174382 0.80 MAPK3 (0.48) KDM4ESMN1; SMN2NSD2ALDH1A1LMNA
SCHEMBL9965412 0.80 MLNR (0.47) KDM4ESMN1; SMN2NSD2ALDH1A1LMNA
SCHEMBL641004 0.79 LMNA (0.65) KDM4ESMN1; SMN2NSD2ALDH1A1LMNA
SCHEMBL2884743 0.78 MAPT (0.43) KDM4ESMN1; SMN2NSD2ALDH1A1LMNA
SCHEMBL641860 0.78 NSD2 (0.51) KDM4ESMN1; SMN2NSD2ALDH1A1KMT2A
SCHEMBL28588875 0.77 MAPT (0.48) NSD2KMT2ABRD4MAPTEPHX2
SCHEMBL30352893 0.77 EPHX2 (0.55) NSD2ALDH1A1KMT2ABRD4MAPT
SCHEMBL643978 0.77 MAPT (0.48) KDM4ESMN1; SMN2NSD2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-B1 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS STERIX LTD (GB) 2012-06-20 EP disclosed