SCHEMBL9965476

SCHEMBL9965476

CC(=O)N1CCC(Nc2ccccc2Cc2ccc(Cl)cc2)CC1c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.42
P2RX7 Q99572 3/20 0.41
SIGMAR1 Q99720 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TACR1 P25103 2/20 0.37
PRCP P42785 1/20 0.37
IDH1 O75874 1/20 0.36
ABCB11 O95342 2/20 0.36
HSD11B1 P28845 1/20 0.36
POLB P06746 1/20 0.36
RIPK1 Q13546 1/20 0.35
FFAR1 O14842 1/20 0.35
APP P05067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965449 0.81 KDM4E (0.51) HRH1SIGMAR1ALDH1A1LMNAKDM4E
SCHEMBL9965463 0.80 EPHX2 (0.40) P2RX7LMNAKDM4ESMN1; SMN2ABCB11
SCHEMBL14639728 0.70 EPHX2 (0.40) TACR1HSD11B1POLBRIPK1
SCHEMBL18711673 0.68 CCNC (0.49) ALDH1A1HSD11B1POLBRIPK1
SCHEMBL24011067 0.67 RIPK1 (0.68) HSD11B1POLBRIPK1
SCHEMBL9965374 0.67 PKM (0.38) ALDH1A1LMNAKDM4EABCB11
SCHEMBL9201806 0.65 TACR1 (0.54) SMN1; SMN2TACR1RIPK1
SCHEMBL9201803 0.65 TACR1 (0.54) SMN1; SMN2TACR1RIPK1
SCHEMBL4242010 0.65 L3MBTL1 (0.56) ALDH1A1LMNASMN1; SMN2IDH1POLB
SCHEMBL643314 0.65 ABCB11 (0.38) LMNAKDM4EABCB11POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-B1 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS STERIX LTD (GB) 2012-06-20 EP disclosed