SCHEMBL9965456

SCHEMBL9965456

O=C(Nc1ccccc1Oc1cc(Cl)cc(Cl)c1)C1CCN(C(=O)C2=CCCC=C2)CC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
ACHE P22303 1/20 0.48
BACE1 P56817 1/20 0.48
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
MGLL Q99685 7/20 0.46
ALDH1A1 P00352 1/20 0.45
TSHR P16473 2/20 0.42
HSD17B10 Q99714 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 3/20 0.41
CYP3A4 P08684 2/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965415 0.84 ACHE (0.68) KMT2AACHEBACE1GAAPKM
SCHEMBL642196 0.83 GAA (0.56) KMT2AACHEBACE1GAAPKM
SCHEMBL9965428 0.81 GAA (0.53) KMT2AACHEBACE1GAAPKM
SCHEMBL10173892 0.80 GAA (0.54) KMT2AACHEBACE1GAAPKM
SCHEMBL9965426 0.79 GAA (0.56) KMT2AACHEBACE1GAAPKM
SCHEMBL9965459 0.79 GAA (0.53) KMT2AACHEBACE1GAAPKM
SCHEMBL10173900 0.79 PTPN1 (0.53) KMT2AACHEBACE1GAAPKM
SCHEMBL641308 0.78 STS (0.55) KMT2AACHEBACE1GAAPKM
SCHEMBL9965453 0.77 POLB (0.51) KMT2AACHEBACE1GAAPKM
SCHEMBL14639717 0.76 GAA (0.49) KMT2AACHEBACE1GAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-B1 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS STERIX LTD (GB) 2012-06-20 EP disclosed