SCHEMBL9967129

SCHEMBL9967129

N#Cc1cnc(N)nc1-c1c[nH]c2ncc(C(F)(F)F)cc12

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 4/20 0.46
CCNA2 P20248 4/20 0.46
CDK2 P24941 4/20 0.46
CDK9 P50750 4/20 0.46
CDK5 Q00535 5/20 0.45
CDK5R1 Q15078 5/20 0.45
ADORA2A P29274 2/20 0.40
ADORA1 P30542 2/20 0.40
CLK1 P49759 6/20 0.40
DYRK1A Q13627 2/20 0.38
CHUK O15111 2/20 0.38
GSK3B P49841 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAP3K11 Q16584 1/20 0.37
NTRK1 P04629 2/20 0.36
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16361467 0.87 CDK2 (0.38) CCNT1CCNA2CDK2CDK9CLK1
SCHEMBL15722335 0.86 CDK2 (0.37) CCNT1CCNA2CDK2CDK9CLK1
SCHEMBL14147359 0.84 CCNT1 (0.50) CCNT1CCNA2CDK2CDK9CDK5
SCHEMBL15722285 0.84 CCNK (0.37) CCNT1CCNA2CDK2CDK9
SCHEMBL11989644 0.84 HSP90AB1 (0.43) CCNT1CCNA2CDK2CDK9CDK5
SCHEMBL27795425 0.84 CDK2 (0.36) CCNT1CCNA2CDK2CDK9CDK5
SCHEMBL14238585 0.84 CDK2 (0.37) CCNT1CCNA2CDK2CDK9CLK1
SCHEMBL11989908 0.84 HSP90AB1 (0.41) CCNT1CCNA2CDK2CDK9CLK1
SCHEMBL11989645 0.83 CDK7 (0.38) CCNT1CCNA2CDK2CDK9CDK5
SCHEMBL9967446 0.82 MAP3K14 (0.48) CCNT1CCNA2CDK2CDK9CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083122-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICAL INCORPORATED (US) 2012-06-21 WO disclosed