SCHEMBL9967204

SCHEMBL9967204

Nc1nc(-c2c[nH]c3ncc(F)cc23)c(C(F)(F)F)cc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.51
CCNT1 O60563 5/20 0.51
CDK9 P50750 5/20 0.51
CCNK O75909 1/20 0.51
CCNE1 P24864 1/20 0.51
CDK12 Q9NYV4 1/20 0.51
CCNA2 P20248 4/20 0.39
GSK3A P49840 6/20 0.38
GSK3B P49841 6/20 0.38
FLT3 P36888 6/20 0.38
PIK3CG P48736 5/20 0.38
CLK1 P49759 4/20 0.38
DYRK1A Q13627 4/20 0.38
PLK1 P53350 4/20 0.38
JAK2 O60674 4/20 0.38
ROCK2 O75116 4/20 0.38
SRC P12931 4/20 0.38
KDR P35968 4/20 0.38
ROCK1 Q13464 4/20 0.38
PIK3CD O00329 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9967235 0.86 CDK2 (0.42) CDK2CCNT1CDK9CCNKCCNE1
SCHEMBL9967124 0.80 KHK (0.42) CDK2CCNT1CDK9CCNKCCNE1
SCHEMBL24840735 0.79 CDK2 (0.57) CDK2CCNT1CDK9CCNKCCNE1
SCHEMBL10304030 0.76 GSK3A (0.53) CDK2GSK3AGSK3BFLT3PIK3CG
SCHEMBL20846287 0.75 CDK2 (0.48) CDK2CCNT1CDK9CCNKCCNE1
SCHEMBL20839192 0.73 CAMKK2 (0.45) CDK2CCNT1CDK9CCNKCCNE1
SCHEMBL9941759 0.72 CDK2 (0.42) CDK2CCNT1CDK9CCNKCCNE1
SCHEMBL24198419 0.72 CLK1 (0.38) CDK2CCNT1CDK9CCNKCCNE1
SCHEMBL25469868 0.72 CCNT1 (0.40) CDK2CCNT1CDK9CCNKCCNE1
SCHEMBL20561594 0.72 CCNT1 (0.44) CDK2CCNT1CDK9CCNKCCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083122-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICAL INCORPORATED (US) 2012-06-21 WO disclosed