SCHEMBL9968636

SCHEMBL9968636

CN1C(=O)C(F)(F)c2c3c(cc(F)c21)N1C(=O)O[C@@H](CNc2ccon2)[C@@H]1C3

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.40
MAOA P21397 2/20 0.36
MAOB P27338 1/20 0.32
CYP2C19 P33261 1/20 0.32
SCN9A Q15858 2/20 0.31
SCN1A P35498 1/20 0.30
SCN5A Q14524 1/20 0.30
SCN8A Q9UQD0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14069265 1.00 CYP2E1 (0.40) CYP2E1MAOAMAOBCYP2C19SCN9A
SCHEMBL9968809 0.89 CYP2E1 (0.40) CYP2E1MAOAMAOBCYP2C19SCN9A
SCHEMBL9968825 0.87 MAOA (0.33) CYP2E1MAOA
SCHEMBL14069618 0.87 MAOA (0.33) CYP2E1MAOA
SCHEMBL9968635 0.84 CYP2E1 (0.41) CYP2E1MAOAMAOBCYP2C19SCN9A
SCHEMBL9968811 0.83 CYP2E1 (0.43) CYP2E1MAOAMAOBCYP2C19SCN9A
SCHEMBL9968808 0.82 CYP2E1 (0.40) CYP2E1MAOAMAOBCYP2C19SCN9A
SCHEMBL9964730 0.81 MAOA (0.49) MAOAMAOBCYP2C19
SCHEMBL14069267 0.80 CYP2E1 (0.39) CYP2E1MAOAMAOBCYP2C19SCN9A
SCHEMBL9968816 0.80 MAOA (0.41) MAOAMAOBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120157434-A1 Antimicrobial heterocyclic compounds for treatment of bacterial infections CSO of MicuRx Pharmaceuticals, Inc. 2012-06-21 US disclosed
WO-2008108988-A1 ANTIMICROBIAL HETEROCYCLIC COMPOUNDS FOR TREATMENT OF BACTERIAL INFECTIONS MICURX PHARMACEUTICALS, INC. (US) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120157434-A1 Antimicrobial heterocyclic compounds for treatment of bacterial infections NISCH, NOD1, NQO1 CYP2E1 144/4885MAOA 1058/4885MAOB 761/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.