SCHEMBL9970824

SCHEMBL9970824

O=C(NC1CCCC(Nc2nc(-c3nn(C(c4ccccc4)(c4ccccc4)c4ccccc4)c4ncc(F)cc34)c(F)cc2F)C1)c1ccsc1Cl

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CDK7 P50613 2/20 0.36
GRM5 P41594 1/20 0.35
HTR3A P46098 4/20 0.33
NR3C1 P04150 1/20 0.33
JAK2 O60674 1/20 0.32
NTRK1 P04629 1/20 0.32
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9970823 0.87 BTK (0.34) CDK7GRM5HTR3A
SCHEMBL15401021 0.84 MAPK3 (0.38) JAK2
SCHEMBL9941262 0.84 MAPK3 (0.38) JAK2
SCHEMBL15400717 0.83 HTR3A (0.34) GRM5HTR3ANTRK1
SCHEMBL9970907 0.80 TP53 (0.37)
SCHEMBL16188366 0.76 PDE5A (0.35) CDK7GRM5
SCHEMBL15400495 0.75 EGFR (0.34)
SCHEMBL9941696 0.73 GSK3A (0.41) JAK2
SCHEMBL9970822 0.73 GSK3A (0.41) JAK2
SCHEMBL15401009 0.73 GSK3A (0.41) JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083121-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-21 WO disclosed