SCHEMBL9970823

SCHEMBL9970823

O=C(NC1CCCC(Nc2nc(-c3nn(C(c4ccccc4)(c4ccccc4)c4ccccc4)c4ncc(F)cc34)c(F)cc2F)C1)c1ccsc1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.34
CDK7 P50613 3/20 0.34
GRM5 P41594 4/20 0.34
HTR3A P46098 1/20 0.32
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9970824 0.87 CDK7 (0.36) CDK7GRM5HTR3A
SCHEMBL15401021 0.85 MAPK3 (0.38) BTK
SCHEMBL9941262 0.85 MAPK3 (0.38) BTK
SCHEMBL15400717 0.85 HTR3A (0.34) BTKGRM5HTR3A
SCHEMBL9970907 0.81 TP53 (0.37)
SCHEMBL9970820 0.81 GRM5 (0.37) BTKCDK7GRM5
SCHEMBL15401564 0.81 GRM5 (0.37) BTKCDK7GRM5
SCHEMBL16188366 0.78 PDE5A (0.35) CDK7GRM5AURKAAURKB
SCHEMBL9967246 0.78 CDK7 (0.43) CDK7
SCHEMBL15400495 0.78 EGFR (0.34) BTKAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083121-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-21 WO disclosed