SCHEMBL9970925

SCHEMBL9970925

Sc1nc(Br)cn2ccnc12

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.44
NUDT1 P36639 1/20 0.36
TNKS O95271 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL103894 0.80 HTR2C (0.53) HTR2CL3MBTL1NUDT1TNKS
SCHEMBL19865160 0.77 L3MBTL1 (0.53) HTR2CL3MBTL1NUDT1TNKS
SCHEMBL24386932 0.77 HTR2C (0.50) HTR2CL3MBTL1NUDT1TNKS
SCHEMBL5477688 0.77 NUDT1 (0.55) HTR2CL3MBTL1NUDT1TNKS
SCHEMBL5405262 0.73 HTR2C (0.47) HTR2CL3MBTL1NUDT1
SCHEMBL2273731 0.73 HTR2C (0.47) HTR2CL3MBTL1NUDT1
SCHEMBL24529236 0.73 HTR2C (0.47) HTR2CL3MBTL1NUDT1TNKS
SCHEMBL24529479 0.73 HTR2C (0.47) HTR2CL3MBTL1NUDT1TNKS
SCHEMBL104884 0.73 HTR2C (0.47) HTR2CL3MBTL1NUDT1TNKS
SCHEMBL1934651 0.73 HTR2C (0.50) HTR2CL3MBTL1NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012080234-A1 SUBSTITUTED 6-IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-21 WO disclosed
WO-2012080228-A1 6-THIO-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-21 WO disclosed