SCHEMBL9974933

SCHEMBL9974933

c1ccc(-c2ccc(-c3cc(-c4ccc(-c5ccccn5)cc4)c(-c4ccc(-c5cncnc5)cc4)cc3-c3ccc(-c4cncnc4)cc3)cc2)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.51
ATM Q13315 1/20 0.47
GRM5 P41594 1/20 0.42
CYP1A2 P05177 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
CCR1 P32246 1/20 0.42
CCR5 P51681 1/20 0.42
CCR8 P51685 1/20 0.42
METAP1 P53582 1/20 0.42
BLM P54132 1/20 0.42
HIF1A Q16665 1/20 0.42
DOHH Q9BU89 1/20 0.42
P4HTM Q9NXG6 1/20 0.42
CHEK2 O96017 1/20 0.42
TGFBR1 P36897 3/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9975012 0.95 CYP2A6 (0.53) CYP2A6ATMGRM5CYP1A2KDM4E
SCHEMBL9975005 0.93 CYP2A6 (0.47) CYP2A6ATMGRM5CYP1A2KDM4E
SCHEMBL14655918 0.86 KDM4E (0.56) CYP2A6CYP1A2KDM4ELMNAPOLB
SCHEMBL9974981 0.85 CYP2A6 (0.69) CYP2A6GRM5CYP1A2TGFBR1CYP19A1
SCHEMBL9974982 0.84 CYP2A6 (0.47) CYP2A6GRM5CYP1A2KDM4ELMNA
SCHEMBL9974919 0.84 LMNA (0.50) CYP2A6CYP1A2KDM4ELMNAPOLB
SCHEMBL9974928 0.83 CYP2A6 (0.71) CYP2A6GRM5CYP1A2KDM4ECHEK2
SCHEMBL9974929 0.82 CYP2A6 (0.48) CYP2A6CYP1A2KDM4ELMNAPOLB
SCHEMBL9974931 0.82 KDM4E (0.52) CYP2A6CYP1A2KDM4ELMNAPOLB
SCHEMBL9974907 0.82 LMNA (0.52) CYP2A6CYP1A2KDM4ELMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012081541-A1 1, 2, 4, 5-SUBSTITUTED PHENYL DERIVATIVE, PRODUCTION METHOD FOR SAME, AND ORGANIC ELECTROLUMINESCENT ELEMENT 東ソー株式会社 (JP) 2012-06-21 WO disclosed