SCHEMBL9977912

SCHEMBL9977912

CCOC(=O)C(=O)Nc1ccc(OC)cc1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.70
ALDH1A1 P00352 6/20 0.69
KDM4E B2RXH2 3/20 0.69
HPGD P15428 1/20 0.69
MAPT P10636 4/20 0.69
NPC1 O15118 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
RAB9A P51151 1/20 0.58
KMT2A Q03164 1/20 0.56
LMNA P02545 1/20 0.55
MAPK1 P28482 1/20 0.55
CYP1A2 P05177 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11408843 0.89 MAPT (0.83) CYP19A1ALDH1A1KDM4EHPGDMAPT
SCHEMBL10987231 0.88 MAPT (0.71) CYP19A1ALDH1A1KDM4EHPGDMAPT
SCHEMBL11510257 0.88 MAPT (0.71) CYP19A1ALDH1A1KDM4EHPGDMAPT
SCHEMBL10557875 0.84 MAPT (0.75) CYP19A1ALDH1A1KDM4EHPGDMAPT
SCHEMBL11608031 0.84 MAPT (0.75) CYP19A1ALDH1A1KDM4EHPGDMAPT
SCHEMBL18415556 0.84 RAB9A (0.68) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL7556396 0.83 NPC1 (0.69) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL626949 0.83 MAPT (0.73) CYP19A1ALDH1A1KDM4EHPGDMAPT
SCHEMBL11536521 0.83 HPGD (0.73) CYP19A1ALDH1A1KDM4EHPGDMAPT
SCHEMBL9674962 0.82 CYP19A1 (0.52) CYP19A1ALDH1A1KDM4EHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3966965-A Oxamic acid derivatives for the prevention of immediate type hypersensitivity reactions AMERICAN HOME PRODUCTS CORPORATION (US) 1976-06-29 US claimed
US-20250092001-A1 NOVEL EXCITATORY AMINO ACID GLUTAMATE TRANSPORT MODULATORS AND METHODS USING THE SAME UNIV DREXEL (US) 2025-03-20 US disclosed
EP-4469440-A1 NOVEL EXCITATORY AMINO ACID GLUTAMATE TRANSPORT MODULATORS AND METHODS USING THE SAME Drexel University (US) 2024-12-04 EP disclosed
CN-118946550-A Novel excitatory amino acid glutamate transport modulators and methods of use thereof 德雷克塞尔大学 2024-11-12 CN disclosed
WO-2023146831-A1 NOVEL EXCITATORY AMINO ACID GLUTAMATE TRANSPORT MODULATORS AND METHODS USING THE SAME DREXEL UNIVERSITY (US) 2023-08-03 WO disclosed
CN-115611793-A Method for synthesizing thioamide compound 山东新华制药股份有限公司 2023-01-17 CN disclosed
US-8546397-B2 DNA methylation inhibitors THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2013-10-01 US disclosed
WO-2012087889-A2 DNA METHYLATION INHIBITORS THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2012-06-28 WO disclosed
US-20120157465-A1 DNA METHYLATION INHIBITORS THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2012-06-21 US disclosed
US-4191840-A Oxamic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1980-03-04 US disclosed
US-4160100-A OXAMIC ACID DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1979-07-03 US disclosed
US-4154961-A Oxamic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1979-05-15 US disclosed
US-4137325-A Antisecretory oxamic acid esters AMERICAN HOME PRODUCTS CORPORATION (US) 1979-01-30 US disclosed
US-4099007-A N,N-SUBSTITUTED 2,4,5-TRIKETOIMIDAZOLIDINES AND A PROCESS FOR THEIR PREPARATION HOECHST AKTIENGESELLSCHAFT (DE) 1978-07-04 US disclosed
US-4069343-A OXAMIC ACID DERIVATIVES FOR THE PREVENTION OF IMMEDIATE TYPE HYPERSENSITIVITY REACTIONS AMERICAN HOME PRODUCTS CORPORATION (US) 1978-01-17 US disclosed
US-4054661-A Pyridyl oxamic acid derivatives and use in the prevention of allergic reactions AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4054657-A Pyrimidinyl oxamic acids and esters, and compositions and methods for the suppression of allergic manifestations AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4054666-A Compositions and methods of treating immediate hypersensitivity reactions with thiazolyl oxamic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4036837-A 2 Alkoxyoxamoyl-pyrazines AMERICAN HOME PRODUCTS CORPORATION (US) 1977-07-19 US disclosed
US-3966965-A Oxamic acid derivatives for the prevention of immediate type hypersensitivity reactions AMERICAN HOME PRODUCTS CORPORATION (US) 1976-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120157465-A1 DNA METHYLATION INHIBITORS MECP2, DNMT1, DNMT3B CYP19A1 1708/4885ALDH1A1 2789/4885KDM4E 427/4885
US-20250092001-A1 NOVEL EXCITATORY AMINO ACID GLUTAMATE TRANSPORT MODULATORS AND METHODS USING THE SAME SLC1A2, SLC1A3, SLC1A1 CYP19A1 4528/4885ALDH1A1 1199/4885KDM4E 2610/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.