SCHEMBL9978274

SCHEMBL9978274

CC(=O)c1ccc(Cl)c(Cl)c1.Cc1ccn[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
NOTUM Q6P988 1/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
PKM P14618 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.41
ALOX15 P16050 1/20 0.41
MAOB P27338 3/20 0.41
MAOA P21397 1/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
OPRK1 P41145 1/20 0.40
TLK2 Q86UE8 1/20 0.40
HPGD P15428 1/20 0.40
F2 P00734 1/20 0.39
PLAU P00749 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL313211 0.80 TSHR (0.64) TSHRNPC1RAB9APKMSMN1; SMN2
SCHEMBL29655535 0.80 TSHR (0.64) TSHRNPC1RAB9APKMSMN1; SMN2
SCHEMBL8478583 0.80 TSHR (0.64) TSHRNPC1RAB9APKMSMN1; SMN2
Nitrogen SCHEMBL28140075 0.76 TSHR (0.59) TSHRNPC1RAB9APKMSMN1; SMN2
Bicarbonate SCHEMBL6567102 0.72 HCAR2 (0.52) NPC1RAB9APKMSMN1; SMN2TP53
Vinyl Chloride SCHEMBL27987346 0.72 TSHR (0.53) TSHRNPC1RAB9APKMSMN1; SMN2
SCHEMBL45219 0.70
SCHEMBL29554593 0.69 MAPT (0.52) TSHRNPC1RAB9APKMSMN1; SMN2
SCHEMBL312135 0.69 MAPT (0.52) TSHRNPC1RAB9APKMSMN1; SMN2
SCHEMBL703716 0.69 HPGD (0.53) NPC1RAB9ASMN1; SMN2POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2576543-A1 PYRAZOLE COMPOUNDS AS SIGMA RECEPTOR INHIBITORS Laboratorios del Dr. Esteve S.A. (ES) 2013-04-10 EP disclosed
WO-2011147910-A1 PYRAZOLE COMPOUNDS AS SIGMA RECEPTOR INHIBITORS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2011-12-01 WO disclosed