SCHEMBL9978669

SCHEMBL9978669

O=C(O)Oc1cc([N+](=O)[O-])n[nH]1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.33
ALOX5 P09917 1/20 0.31
LMNA P02545 2/20 0.30
TDP1 Q9NUW8 2/20 0.30
F2 P00734 1/20 0.30
PLAU P00749 1/20 0.30
KLKB1 P03952 1/20 0.30
ELANE P08246 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
AHR P35869 1/20 0.30
RAB9A P51151 1/20 0.30
CASP6 P55212 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
GRK6 P43250 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27683380 0.85 DYRK1A (0.34)
SCHEMBL6167693 0.82 DYRK1A (0.35) MEN1POLBKMT2AL3MBTL1
SCHEMBL28802178 0.77 MAPT (0.36) SMN1; SMN2LMNATDP1MEN1RAB9A
SCHEMBL160276 0.73 SMN1; SMN2 (0.51) SMN1; SMN2
SCHEMBL377046 0.72 HCAR2 (0.32)
SCHEMBL16524045 0.71 SMN1; SMN2 (0.37) SMN1; SMN2LMNAMEN1POLBKMT2A
SCHEMBL6169307 0.71 DYRK1A (0.33) SMN1; SMN2MEN1KMT2A
Water SCHEMBL7303697 0.71 HCAR2 (0.32)
SCHEMBL3931686 0.71 HCAR2 (0.38)
SCHEMBL10399828 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3747454-B9 AMYLOID-BETA BINDING PEPTIDES AND THESE PEPTIDES FOR USE IN THE THERAPY AND DIAGNOSIS OF ALZHEIMER'S DEMENTIA PRIAVOID GMBH (DE) 2023-10-04 EP disclosed
EP-3747454-B1 AMYLOID-BETA BINDING PEPTIDES AND THESE PEPTIDES FOR USE IN THE THERAPY AND DIAGNOSIS OF ALZHEIMER'S DEMENTIA PRIAVOID GMBH (DE) 2023-06-07 EP disclosed
EP-3346273-B1 NOVEL D-ENANTIOMERIC PEPTIDES DERIVED FROM D3 AND THEIR USE PRIAVOID GMBH (DE) 2023-01-04 EP disclosed
EP-3747454-A1 AMYLOID-BETA BINDING PEPTIDES AND THEIR USE IN THE THERAPY AND DIAGNOSIS OF ALZHEIMER'S DEMENTIA Forschungszentrum Jülich GmbH (DE) 2020-12-09 EP disclosed
EP-3049099-B1 AMYLOID-BETA-BINDING PEPTIDES AND THE USE THEREOF FOR THE THERAPY AND DIAGNOSIS OF ALZHEIMER'S DEMENTIA FORSCHUNGSZENTRUM JUELICH GMBH (DE) 2020-06-17 EP disclosed
EP-3271374-B1 PEPTIDES WHICH BIND TO A SPECIFIC A-BETA-SPECIES FOR THE THERAPY AND/OR DIAGNOSIS OF ALZHEIMER'S DISEASE FORSCHUNGSZENTRUM JUELICH GMBH (DE) 2020-06-03 EP disclosed
EP-3558336-A1 D-ENANTIOMERIC PEPTIDES FOR THE THERAPY OF CHRONIC AND NEUROPATHIC PAIN Forschungszentrum Jülich GmbH (DE) 2019-10-30 EP disclosed
EP-2895867-B1 NOVEL D-ENANTIOMERIC PEPTIDES DERIVED FROM D3 AND USE THEREOF FORSCHUNGSZENTRUM JUELICH GMBH (DE) 2019-10-23 EP disclosed
EP-3296316-B1 PEPTIDES FOR THE TREATMENT AND EARLY DIAGNOSIS OF ALZHEIMER'S DISEASE AND OTHER TAUOPATHIES FORSCHUNGSZENTRUM JUELICH GMBH (DE) 2019-05-22 EP disclosed
EP-3296315-B1 PEPTIDES FOR THE TREATMENT AND EARLY DIAGNOSIS OF ALZHEIMER'S DISEASE AND OTHER TAUOPATHIES FORSCHUNGSZENTRUM JUELICH GMBH (DE) 2019-05-08 EP disclosed
EP-3271374-A1 PEPTIDES WHICH BIND TO A SPECIFIC A-BETA-SPECIES FOR THE THERAPY AND/OR DIAGNOSIS OF ALZHEIMER'S DISEASE Forschungszentrum Jülich GmbH (DE) 2018-01-24 EP disclosed
WO-2016150415-A1 PEPTIDES WHICH BIND TO A SPECIFIC A-BETA-SPECIES FOR THE THERAPY AND/OR DIAGNOSIS OF ALZHEIMER'S DISEASE Forschungszentrum Jülich GmbH (DE) 2016-09-29 WO disclosed
WO-2016150416-A1 SPECIFIC AMYLOID BETA BINDING PEPTIDES AND THE USE OF SAME FOR TREATING AND DIAGNOSING ALZHEIMER'S DEMENTIA Forschungszentrum Jülich GmbH (DE) 2016-09-29 WO disclosed
EP-3049099-A1 AMYLOID-BETA-BINDING PEPTIDES AND THE USE THEREOF FOR THE THERAPY AND DIAGNOSIS OF ALZHEIMER'S DEMENTIA Forschungszentrum Jülich GmbH (DE) 2016-08-03 EP disclosed
EP-2903999-A2 PEPTIDES FOR THE TREATMENT AND EARLY DIAGNOSIS OF ALZHEIMER'S DISEASE AND OTHER TAUOPATHIES Forschungszentrum Jülich Gmbh (DE) 2015-08-12 EP disclosed
EP-2895867-A2 NOVEL D-ENANTIOMERIC PEPTIDES DERIVED FROM D3 AND USE THEREOF Forschungszentrum Jülich Gmbh (DE) 2015-07-22 EP disclosed
WO-2015043567-A1 AMYLOID-BETA-BINDING PEPTIDES AND THE USE THEREOF FOR THE THERAPY AND DIAGNOSIS OF ALZHEIMER'S DEMENTIA Forschungszentrum Jülich GmbH (DE) 2015-04-02 WO disclosed
WO-2014053110-A2 PEPTIDES FOR THE TREATMENT AND EARLY DIAGNOSIS OF ALZHEIMER'S DISEASE AND OTHER TAUOPATHIES Forschungszentrum Jülich GmbH (DE) 2014-04-10 WO disclosed
WO-2014041115-A2 NOVEL D-ENANTIOMERIC PEPTIDES DERIVED FROM D3 AND USE THEREOF Forschungszentrum Jülich GmbH (DE) 2014-03-20 WO disclosed
WO-2011147797-A2 HYBRID COMPOUND, THE USE THEREOF, AND METHOD FOR THE PRODUCTION THEREOF Forschungszentrum Jülich GmbH (DE) 2011-12-01 WO disclosed