SCHEMBL9986241

SCHEMBL9986241

C[C@@]1(c2cc(F)cc(F)c2)CN(C(=O)O)C2(CCCCCC2)C(=O)N1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.38
HCAR3 P49019 1/20 0.38
OPRM1 P35372 2/20 0.32
SLC6A9 P48067 2/20 0.32
RIPK1 Q13546 1/20 0.32
CALCRL Q16602 1/20 0.31
ADAMTS5 Q9UNA0 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL979071 1.00 HCAR2 (0.38) HCAR2HCAR3OPRM1SLC6A9RIPK1
SCHEMBL981294 0.99 HCAR2 (0.39) HCAR2HCAR3OPRM1SLC6A9RIPK1
SCHEMBL979177 0.84 GRIN2B (0.35) HCAR2HCAR3HDAC1HDAC2
SCHEMBL12948254 0.83 GRIN2B (0.36) HCAR2HCAR3OPRM1HDAC1HDAC2
SCHEMBL12028357 0.81 CALCRL (0.36) HCAR2HCAR3OPRM1SLC6A9CALCRL
SCHEMBL5654621 0.77 HDAC4 (0.41) HCAR2HCAR3OPRM1SLC6A9HDAC3
SCHEMBL979178 0.72 HCAR3 (0.35) HCAR2HCAR3OPRM1SLC6A9
SCHEMBL978532 0.71 KMT2A (0.30)
SCHEMBL12028354 0.71 S1PR1 (0.31) HCAR2HCAR3HDAC3HDAC1HDAC2
SCHEMBL1273276 0.71 HDAC4 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8507477-B2 3- and 6-quinolines with N-attached heterocyclic CGRP receptor antagonists Merck, Sharp & Dohme, Corp. (US) 2013-08-13 US disclosed
US-20110306604-A1 3- AND 6-QUINOLINES WITH N-ATTACHED HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LLC 2011-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110306604-A1 3- AND 6-QUINOLINES WITH N-ATTACHED HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS CALCRL, CCKBR, CCKAR HCAR2 83/4885HCAR3 24/4885OPRM1 73/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.