SCHEMBL9987333

SCHEMBL9987333

COc1ccc(COc2nc(Cl)ncc2C(C)C)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.44
APP P05067 7/20 0.43
CNR2 P34972 3/20 0.42
CNR1 P21554 2/20 0.42
PIN1 Q13526 1/20 0.41
HRH4 Q9H3N8 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
IDO1 P14902 1/20 0.39
AGXT P21549 1/20 0.39
BCHE P06276 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
PDE2A O00408 1/20 0.39
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9987222 0.83 CNR1 (0.44) MAOBAPPCNR2CNR1PIN1
SCHEMBL22323930 0.82 APP (0.50) MAOBAPPCNR2CNR1PIN1
SCHEMBL3196355 0.82 CNR1 (0.43) MAOBAPPCNR2CNR1PIN1
SCHEMBL846643 0.82 POLB (0.47) MAOBAPPCNR2CNR1PIN1
SCHEMBL31514820 0.82 CNR1 (0.43) MAOBAPPCNR2CNR1PIN1
SCHEMBL9987933 0.81 PIN1 (0.44) MAOBAPPCNR2CNR1PIN1
SCHEMBL20564303 0.80 MAOB (0.43) MAOBAPPCNR2CNR1HRH4
SCHEMBL20565236 0.78 AR (0.43) MAOBAPPCNR2CNR1PIN1
SCHEMBL20564322 0.78 CNR2 (0.43) MAOBAPPCNR2CNR1HRH4
SCHEMBL20564007 0.77 HTR6 (0.40) MAOBAPPCNR2CNR1PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011158149-A1 2-(3,5-DISUBSTITUTEDPHENYL)PYRIMIDIN-4(3H)-ONE DERIVATIVES PFIZER INC. (US) 2011-12-22 WO disclosed
WO-2011158149-A1 2-(3,5-DISUBSTITUTEDPHENYL)PYRIMIDIN-4(3H)-ONE DERIVATIVES PFIZER INC. (US) 2011-12-22 WO disclosed