SCHEMBL9987584

SCHEMBL9987584

CC(C)Nc1ccc([N+](=O)[O-])c(Nc2ccc(N3CCC(C(=O)O)CC3)c(F)c2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 7/20 0.51
TDP1 Q9NUW8 1/20 0.46
NTRK1 P04629 1/20 0.41
SERPINE1 P05121 2/20 0.40
JAK2 O60674 1/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 4/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
POLB P06746 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.38
RET P07949 1/20 0.38
ROS1 P08922 1/20 0.38
FLT3 P36888 1/20 0.38
EML4 Q9HC35 1/20 0.38
ALK Q9UM73 1/20 0.38
RHOA P61586 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9984137 0.92 BRD4 (0.50) BRD4NTRK1MAPTMAPK1POLB
SCHEMBL9984423 0.91 BRD4 (0.53) BRD4NTRK1KMT2AMAPTMEN1
SCHEMBL9987376 0.91 TDP1 (0.48) BRD4TDP1SERPINE1JAK2KMT2A
SCHEMBL9987060 0.89 TDP1 (0.43) BRD4TDP1SERPINE1JAK2KMT2A
SCHEMBL9983765 0.89 BRD4 (0.53) BRD4NTRK1MAPTMAPK1CYP2C9
SCHEMBL9984854 0.88 BRD4 (0.57) BRD4NTRK1MAPTMAPK1CYP2C9
SCHEMBL9987013 0.86 TDP1 (0.39) BRD4TDP1SERPINE1JAK2RET
SCHEMBL9984657 0.85 BRD4 (0.48) BRD4NTRK1KMT2AMAPTMEN1
SCHEMBL9984381 0.85 BRD4 (0.57) BRD4NTRK1MAPTMAPK1GAA
SCHEMBL9985174 0.85 BRD4 (0.55) BRD4NTRK1MAPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394993-A2 NOVEL 2,6-SUBSTITUTED-3-NITROPYRIDINE DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION INCLUDING SAME Dong Wha Pharm. Co., Ltd. (KR) 2011-12-14 EP disclosed