SCHEMBL9987666

SCHEMBL9987666

CCOC(=O)n1nc(Br)c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.55
F2 P00734 1/20 0.52
PLAU P00749 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5120293 0.86 ELANE (0.56) ELANEF2PLAU
SCHEMBL5120296 0.83 ELANE (0.56) ELANEF2PLAU
SCHEMBL517483 0.82 ELANE (0.55) ELANEF2PLAU
SCHEMBL2674135 0.81 MAP2K4 (0.44) ELANEF2PLAU
SCHEMBL6852832 0.81 ELANE (0.53) ELANEF2PLAU
SCHEMBL4753928 0.80 ELANE (0.50) ELANEF2PLAU
SCHEMBL11753223 0.79 ELANE (0.52) ELANEF2PLAU
SCHEMBL5583818 0.79 ELANE (0.54) ELANEF2PLAU
SCHEMBL25769987 0.77 ELANE (0.40) ELANEF2PLAU
SCHEMBL5109043 0.75 ELANE (0.48) ELANEF2PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2584903-A1 NOVEL HETEROCYCLIC COMPOUNDS AS ERK INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-01 EP disclosed
WO-2011163330-A1 NOVEL HETEROCYCLIC COMPOUNDS AS ERK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-12-29 WO disclosed