SCHEMBL9989075

SCHEMBL9989075

COC(=O)N1C[CH]C[C@@H](OC)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.42
CHRNA4 P43681 2/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
TSHR P16473 1/20 0.38
PDE4B Q07343 5/20 0.35
PDE4A P27815 3/20 0.35
PDE4C Q08493 3/20 0.35
PDE4D Q08499 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
USP2 O75604 1/20 0.33
KMT2A Q03164 3/20 0.32
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
KIF11 P52732 1/20 0.31
MEN1 O00255 2/20 0.30
CYP3A4 P08684 1/20 0.30
MAPK1 P28482 1/20 0.30
CYP2C19 P33261 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9987915 0.83 CHRNB2 (0.35) CHRNB2CHRNA4CHRNB4CHRNA3PDE4B
SCHEMBL19686899 0.80 CHRNB2 (0.55) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL20240587 0.77 JAK3 (0.40) KMT2A
SCHEMBL4277569 0.75
SCHEMBL19686581 0.73 CHRNB2 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL9987717 0.73 CHRNB2 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL791909 0.73 CHRNB2 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL26793108 0.73 CHRNB2 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL791935 0.70 PDE4B (0.43) CHRNB2CHRNA4CHRNB4CHRNA3TSHR
SCHEMBL31107954 0.70 PREP (0.44) PDE4BL3MBTL1USP2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2397462-A2 Compounds, compositions and methods of treatment for heart failure Cytokinetics, Inc. (US) 2011-12-21 EP disclosed