SCHEMBL9995773

SCHEMBL9995773

CC(O)CNCCCCS(=O)(=O)CCCC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.40
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
CES1 P23141 5/20 0.33
MEN1 O00255 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SLC2A1 P11166 1/20 0.32
FAAH O00519 3/20 0.30
CES2 O00748 2/20 0.30
TDP1 Q9NUW8 1/20 0.30
MAPK1 P28482 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9995602 1.00 PKM (0.40) PKMKDM4EALDH1A1GAACES1
SCHEMBL9995784 1.00 PKM (0.40) PKMKDM4EALDH1A1GAACES1
SCHEMBL9995708 0.78 CA3 (0.34) CES1FAAHCES2
SCHEMBL9995669 0.75 CES1 (0.33) CES1FAAHCES2
SCHEMBL918439 0.73 KMT2A (0.38) PKMKDM4EALDH1A1GAAMEN1
SCHEMBL918428 0.73 KMT2A (0.38) PKMKDM4EALDH1A1GAAMEN1
SCHEMBL918429 0.73 KMT2A (0.38) PKMKDM4EALDH1A1GAAMEN1
SCHEMBL9995593 0.72 CA3 (0.32)
SCHEMBL309951 0.72 CES1 (0.33) CES1FAAHCES2
SCHEMBL14775056 0.70 CES1 (0.36) CES1FAAHCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585435-A1 6,7-DIHYDRO-5H-BENZO[7]ANNULENE DERIVATIVES, PROCESS FOR PREPARATION THEREOF, PHARMACEUTICAL PREPARATIONS COMPRISING THEM, AND THE USE THEREOF FOR PRODUCTION OF MEDICAMENTS Bayer Intellectual Property GmbH (DE) 2013-05-01 EP disclosed
WO-2011161101-A1 6,7-DIHYDRO-5H-BENZO[7]ANNULENE DERIVATIVES, PROCESS FOR PREPARATION THEREOF, PHARMACEUTICAL PREPARATIONS COMPRISING THEM, AND THE USE THEREOF FOR PRODUCTION OF MEDICAMENTS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-12-29 WO disclosed