SCHEMBL9995992

SCHEMBL9995992

O=C(O)Oc1cc(Cn2nnc(C(F)(F)F)n2)nn1-c1ncccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.36
TRPV1 Q8NER1 1/20 0.36
SLC16A3 O15427 16/20 0.35
SLC16A1 P53985 15/20 0.35
MCTS1 Q9ULC4 9/20 0.35
DHODH Q02127 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2490874 0.91 SLC16A3 (0.34) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL2134837 0.86 NPC1 (0.35) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL45281 0.85 TRPA1 (0.35) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL45189 0.84 TRPA1 (0.34) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL2491219 0.84 TRPA1 (0.33) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL24287198 0.84 TRPA1 (0.34) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL30388183 0.83 SCN9A (0.36) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL2623668 0.83 DHODH (0.36) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL16530247 0.83 TRPA1 (0.35) TRPA1TRPV1SLC16A3SLC16A1MCTS1
SCHEMBL16014772 0.82 SLC16A3 (0.38) TRPA1TRPV1SLC16A3SLC16A1MCTS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2955176-B1 COMPOSITION COMPRISING CRYSTALLINE FORM B OF 1- (3-CHLOROPYRIDIN-2-YL)-N-[4-CYANO-2-METHYL-6-(METHYLCARBAMOYL)PHENYL]-3-([5-(TRIFLUOROMETHYL)-2H- TETRAZOL-2-YL]METHYL)-1H-PYRAZOL-5-CARBOXAMIDE AND ITS USE BAYER IP GMBH (DE) 2017-12-06 EP disclosed
EP-2955176-A1 COMPOSITION COMPRISING CRYSTALLINE FORM B of 1- (3-CHLOROPYRIDIN-2-YL)-N-[4-CYANO-2-METHYL-6-(METHYLCARBAMOYL)PHENYL]-3-{[5-(TRIFLUOROMETHYL)-2H- TETRAZOL-2-YL]METHYL}-1H-PYRAZOL-5-CARBOXAMIDE AND ITS USE Bayer Intellectual Property GmbH (DE) 2015-12-16 EP disclosed
EP-2582694-B1 PROCESS FOR MANUFACTURING TETRAZOLE- SUBSTITUTED ANTHRANILIC ACID DIAMIDE DERIVATIVES AND NOVEL CRYSTALLINE MODIFICATION OF THESE DERIVATIVES BAYER IP GMBH (DE) 2015-07-22 EP disclosed
EP-2582694-A1 PROCESS FOR PREPARING TETRAZOLE-SUBSTITUTED ANTHRANILAMIDE DERIVATIVES AND NOVEL CRYSTAL POLYMORPH OF THESE DERIVATIVES Bayer Intellectual Property GmbH (DE) 2013-04-24 EP disclosed
WO-2011157664-A1 PROCESS FOR PREPARING TETRAZOLE-SUBSTITUTED ANTHRANILAMIDE DERIVATIVES AND NOVEL CRYSTAL POLYMORPH OF THESE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2011-12-22 WO disclosed