SCHEMBL9998541

SCHEMBL9998541

CC(=O)OC/C(=C\c1cccc(Br)c1)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.41
ALDH1A1 P00352 3/20 0.41
HCAR2 Q8TDS4 1/20 0.40
PLAAT5 Q96KN8 1/20 0.40
PLAAT4 Q9UL19 1/20 0.40
MAPT P10636 2/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
EGFR P00533 1/20 0.39
ERBB2 P04626 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
HSD17B3 P37058 1/20 0.38
SLC6A19 Q695T7 1/20 0.38
POLB P06746 1/20 0.38
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9998543 1.00 PKM (0.41) PKMALDH1A1HCAR2PLAAT5PLAAT4
SCHEMBL9997388 0.87 ALDH1A1 (0.50) ALDH1A1AKR1C3CYP3A4CYP2C9
SCHEMBL9997387 0.87 ALDH1A1 (0.50) ALDH1A1AKR1C3CYP3A4CYP2C9
SCHEMBL9997493 0.86 ALDH1A1 (0.42) PKMALDH1A1MAPTCYP3A4CYP2C9
SCHEMBL9998527 0.86 ALDH1A1 (0.42) ALDH1A1MAPTCYP3A4CYP2C9POLB
SCHEMBL9998528 0.86 ALDH1A1 (0.42) ALDH1A1MAPTCYP3A4CYP2C9POLB
SCHEMBL9997492 0.86 ALDH1A1 (0.42) PKMALDH1A1MAPTCYP3A4CYP2C9
SCHEMBL9997518 0.86 ALDH1A1 (0.44) ALDH1A1MAPTAKR1C3EGFRERBB2
SCHEMBL9997520 0.86 ALDH1A1 (0.44) ALDH1A1MAPTAKR1C3EGFRERBB2
SCHEMBL9997433 0.85 KMT2A (0.44) PKMALDH1A1HCAR2MAPTAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8558012-B2 2-fluoro-1,3-benzodithiol 1,1,3,3-tetraoxide derivative, production method thereof, and production method of monofluoromethyl group-containing compound using the same NAGOYA INSTITUTE OF TECHNOLOGY (JP) 2013-10-15 US disclosed
US-20110319637-A1 2-FLUORO-1,3-BENZODITHIOL 1,1,3,3-TETRAOXIDE DERIVATIVE, PRODUCTION METHOD THEREOF, AND PRODUCTION METHOD OF MONOFLUOROMETHYL GROUP-CONTAINING COMPOUND USING THE SAME NAGOYA INSTITUTE OF TECHNOLOGY (JP) 2011-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110319637-A1 2-FLUORO-1,3-BENZODITHIOL 1,1,3,3-TETRAOXIDE DERIVATIVE, PRODUCTION METHOD THEREOF, AND PRODUCTION METHOD OF MONOFLUOROMETHYL GROUP-CONTAINING COMPOUND USING THE SAME CBR1, CYP1B1, CYP2F1 PKM 1948/4885ALDH1A1 160/4885HCAR2 1256/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.