SCHEMBL1000536

SCHEMBL1000536

C=C(CBr)C1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
EPHX1 P07099 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
NOS2 P35228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1000511 0.97
SCHEMBL19047399 0.86
SCHEMBL3605682 0.76 CES2 (0.39) MGLLCES2CES1HDAC8HDAC6
SCHEMBL13652381 0.75 GABRA1 (0.41) TSHRNOS2
SCHEMBL23547192 0.74 CES2 (0.38) MGLLCES2CES1HDAC8HDAC6
SCHEMBL11210860 0.74 CES2 (0.38) MGLLCES2CES1HDAC8HDAC6
SCHEMBL11211286 0.74 CES2 (0.38) MGLLCES2CES1HDAC8HDAC6
SCHEMBL8464246 0.74 CES2 (0.38) MGLLCES2CES1HDAC8HDAC6
SCHEMBL951792 0.72 CES2 (0.36) MGLLCES2CES1HDAC8HDAC6
Hydrochloric Acid SCHEMBL29945534 0.72 CES2 (0.36) MGLLCES2CES1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007396-B1 Enfumafungin derivatives as antifungal agents MERCK SHARP & DOHME (US) 2013-02-13 EP disclosed
EP-2346332-A1 PYRIDO (4,3-B) INDOLES CONTAINING RIGID MOIETIES Medivation Technologies, Inc. (US) 2011-07-27 EP disclosed
US-7863465-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2011-01-04 US disclosed
WO-2010051501-A1 PYRIDO (4,3-B) INDOLES CONTAINING RIGID MOIETIES MEDIVATION TECHNOLOGIES, INC. (US) 2010-05-06 WO disclosed
EP-2007396-A1 ANTIFUNGAL AGENTS Merck and Co., Inc. (US) 2008-12-31 EP disclosed
US-20080009504-A1 Antifungal agents SCYNEXIS, INC. 2008-01-10 US disclosed
WO-2007127012-A1 ANTIFUNGAL AGENTS MERCK & CO., INC. (US) 2007-11-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080009504-A1 Antifungal agents DPM1, MAN2B1, MAN2A1 MGLL 1627/4885CES2 3273/4885CES1 399/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.