SCHEMBL10028023

SCHEMBL10028023

CNCCN1C(=O)CC(C)C1=O

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 2/20 0.36
PRMT6 Q96LA8 2/20 0.36
PRMT8 Q9NR22 2/20 0.36
PRMT1 Q99873 1/20 0.36
CYP19A1 P11511 5/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 3/20 0.32
GAA P10253 2/20 0.31
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15944143 0.89 SLC6A2 (0.38) CYP19A1SMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL16174529 0.88 CYP19A1 (0.38) CYP19A1SMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL16174528 0.86 CYP19A1 (0.39) CYP19A1SMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL14589097 0.84 CYP19A1 (0.39) CYP19A1SMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL16174526 0.84 MGLL (0.33) ALDH1A1
SCHEMBL27269423 0.82 MGLL (0.35) ALDH1A1
SCHEMBL13071687 0.82 CYP19A1 (0.35) PRMT6CYP19A1SMN1; SMN2MEN1KMT2A
SCHEMBL12754941 0.81
SCHEMBL23369332 0.81 CYP19A1 (0.37) CYP19A1SMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL19981935 0.81 ALDH1A1 (0.32) CYP19A1SMN1; SMN2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 52 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023118599-A1 IMPLANTABLE DEVICE COMPRISING A HYDROGEL ADOCIA (FR) 2023-06-29 WO disclosed
EP-4190361-A1 POLYETHYLENE GLYCOL CONJUGATE DRUG, AND PREPARATION METHOD THERFOR AND USE THEREOF Chongqing Upgra Biotechnology Co., Ltd. (CN) 2023-06-07 EP disclosed
EP-4190360-A1 POLYETHYLENE GLYCOL CONJUGATE DRUG SYNERGIST, PREPARATION METHOD THEREFOR, AND USE THEREOF Chongqing Upgra Biotechnology Co., Ltd. (CN) 2023-06-07 EP disclosed
WO-2022148887-A1 HYDROGELS FOR CELL THERAPY ADOCIA (FR) 2022-07-14 WO disclosed
WO-2022022360-A1 POLYETHYLENE GLYCOL CONJUGATE DRUG, AND PREPARATION METHOD THERFOR AND USE THEREOF 重庆阿普格雷生物科技有限公司 2022-02-03 WO disclosed
EP-3313884-B9 ANTI-CD123 ANTIBODIES AND CONJUGATES AND DERIVATIVES THEREOF IMMUNOGEN INC (US) 2021-05-19 EP disclosed
EP-3313884-B1 ANTI-CD123 ANTIBODIES AND CONJUGATES AND DERIVATIVES THEREOF IMMUNOGEN INC (US) 2020-11-18 EP disclosed
WO-2020223351-A1 THERAPEUTIC COMBINATIONS COMPRISING ANTI-CD123 IMMUNOCONJUGATES IMMUNOGEN, INC. (US) 2020-11-05 WO disclosed
WO-2018119196-A1 IMMUNOCONJUGATES TARGETING ADAM9 AND METHODS OF USE THEREOF IMMUNOGEN, INC. (US) 2018-06-28 WO disclosed
US-20170029514-A1 ANTI-CD123 ANTIBODIES AND CONJUGATES AND DERIVATIVES THEREOF IMMUNOGEN, INC. 2017-02-02 US disclosed
US-20090017004-A1 POLYMERIC DRUG DELIVERY SYSTEMS CONTAINING AN AROMATIC ALLYLIC ACID ENZON PHARMACEUTICALS, INC. (US) 2009-01-15 US disclosed
US-20090017004-A1 POLYMERIC DRUG DELIVERY SYSTEMS CONTAINING AN AROMATIC ALLYLIC ACID ENZON PHARMACEUTICALS, INC. (US) 2009-01-15 US disclosed
WO-2009009712-A1 POLYMERIC DRUG DELIVERY SYSTEM CONTAINING A MULTI-SUBSTITUTED AROMATIC MOIETY ENZON PHARMACEUTICALS, INC. (US) 2009-01-15 WO disclosed
WO-2008070477-A9 POLYMERIC SHORT INTERFERING RNA CONJUGATES ENZON PHARMACEUTICALS INC (US) 2008-07-24 WO disclosed
WO-2008034123-A2 POLYMERIC CONJUGATES CONTAINING POSITIVELY-CHARGED MOIETIES ENZON PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed
WO-2008034122-A2 HINDERED ESTER-BASED BIODEGRADABLE LINKERS FOR OLIGONUCLEOTIDE DELIVERY ENZON PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed
WO-2008034124-A2 TARGETED POLYMERIC PRODRUGS CONTAINING MULTIFUNCTIONAL LINKERS ENZON PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed
WO-2008034119-A2 POLYALKYLENE OXIDES HAVING HINDERED ESTER-BASED BIODEGRADABLE LINKERS ENZON PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed
WO-2008034120-A2 LYSINE-BASED POLYMERIC LINKERS ENZON PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed
EP-0867190-B1 CYTOTOXIN COMPLEXES COMPRISING DIPEPTIDES KYOWA HAKKO KOGYO KK (JP) 2007-12-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090017004-A1 POLYMERIC DRUG DELIVERY SYSTEMS CONTAINING AN AROMATIC ALLYLIC ACID AADAC, ACSS2, ANXA6 CARM1 2622/4885PRMT6 1990/4885PRMT8 3316/4885
US-20170029514-A1 ANTI-CD123 ANTIBODIES AND CONJUGATES AND DERIVATIVES THEREOF IL23R, CD22, IL2RA CARM1 3407/4885PRMT6 3305/4885PRMT8 3266/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.