SCHEMBL10028158

SCHEMBL10028158

Fc1ccccc1-c1ccc2cc3oc4ccc5c6cc(-c7ccccc7F)ccc6cc6oc7ccc(c2c1)c3c7-c4c65

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.41
MAP4K4 O95819 1/20 0.40
BACE1 P56817 1/20 0.39
PTPRC P08575 1/20 0.37
PTPN1 P18031 1/20 0.37
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
TRPA1 O75762 1/20 0.36
CYP1A1 P04798 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP1B1 Q16678 2/20 0.36
PRKDC P78527 1/20 0.36
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35
EPHX2 P34913 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
ACMSD Q8TDX5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10028145 0.86 WEE1 (0.40) AHRCYP1A1CYP1A2CYP1B1NPC1
SCHEMBL10028151 0.84 CTSD (0.39) BACE1TRPA1CYP1A2NPC1HPGD
SCHEMBL10028146 0.84 MCL1 (0.38) AHRCYP1A1CYP1A2CYP1B1ACMSD
SCHEMBL10028239 0.74 AHR (0.46) AHRCYP1A1CYP1A2CYP1B1NPC1
SCHEMBL10028107 0.71 GSTP1 (0.44) AHRCYP1A1CYP1A2CYP1B1HDAC8
SCHEMBL31658899 0.70 HPGD (0.51) AHRMAP4K4PTPRCPTPN1TNKS
SCHEMBL10028152 0.68 KDM4E (0.38) AHRCYP1A2
SCHEMBL26750985 0.67 NPC1 (0.48) AHRMAP4K4PTPRCPTPN1TNKS
SCHEMBL10028089 0.67 AHR (0.37) AHRCYP1A1CYP1A2CYP1B1NPC1
SCHEMBL4567313 0.66 TDP1 (0.43) AHRCYP1A1CYP1A2NPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046915-B1 NEW MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2015-12-02 EP disclosed
US-8114531-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2012-02-14 US disclosed
US-8114531-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2012-02-14 US disclosed
US-20100013381-A1 NOVEL MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2010-01-21 US disclosed
US-20100013381-A1 NOVEL MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2010-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100013381-A1 NOVEL MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES L1CAM, SOD1, SLC40A1 AHR 2429/4885MAP4K4 3255/4885BACE1 2454/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.